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(2S,4S)-4-(4-cyanobenzamido)-N-ethyl-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
N-[1-(4-chlorophenyl)ethyl]-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
ethyl 2-{9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl}acetate
methyl 1-[2-(4-fluorophenyl)-3-oxopiperazine-1-carbonyl]cyclopropane-1-carboxylate
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
N5-tert-butyl-N3-methyl-4-oxo-1-(propan-2-yl)-N3-(quinolin-5-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(dimethylamino)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(3-methylphenyl)acetamide
2-[3-(3-acetamidophenyl)phenoxy]propanamide
2-{4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]morpholin-3-yl}acetic acid
4-{6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-1λ6-thiane-1,1-dione
methyl 1-(3-methylbutoxy)-8-[(6-methylpyridin-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N4-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-methylpyrimidine-2,4-diamine
2-({4-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
(4aS,8aS)-2-(6,8-dimethylquinolin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-4-(pyridin-2-yl)piperazine
1-(4,6-dimethylquinazolin-2-yl)-N-[2-(thiophen-2-yl)ethyl]piperidin-4-amine
4-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperazine-2-carboxylic acid
(5S,9aS,9bS)-5-[4-(cyclopentyloxy)phenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanamine
3-({4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]piperidin-1-yl}methyl)phenol
9-(3-chloro-2-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-benzyl-4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-1,4-diazepan-6-ol
2-{1-benzyl-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)imidazolidin-2-one
5-methoxy-2-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]-1,4-dihydropyridin-4-one
N-(5-cyanopyridin-2-yl)-4-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]benzamide
4-(4-fluorophenyl)-1-(5-methylpyrimidin-2-yl)piperidin-4-ol
5-(3-fluorophenoxymethyl)-N-[1-(furan-2-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}azepane
2-(4-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}phenoxy)pyrimidine
4-(4-{[(5-amino-1H-1,2,4-triazol-3-yl)methyl]amino}piperidin-1-yl)-6-ethyl-N,N-dimethylpyrimidin-2-amine
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
6-[(3-hydroxy-4-methoxyphenyl)methyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
3-({7-oxo-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-5-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1-(pyrimidin-2-yl)piperidin-4-amine
N-{1-[1-(3-methylbutyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(1,2-benzoxazol-3-yl)-N-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}acetamide
{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-propylpiperidin-3-yl}methanol
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-4-ol
1-cyclopropyl-5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]piperidin-2-one
2-(1H-1,3-benzodiazol-2-yl)-N-(1-ethyl-3-methyl-1H-pyrazol-4-yl)piperidine-1-carboxamide
1-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
1-[2-(methylsulfanyl)ethyl]-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
N-[2-(2,4-difluorophenyl)-1-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}ethyl]-N-methylcyclopropanecarboxamide
3-({5-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
(2S,4R)-4-{[(2,4-difluorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
N'-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-N,N-dimethylbutanediamide