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1,4-dimethyl-3-(3,4,5-trimethoxyphenyl)-1H-indazole
1-cyclopropanecarbonyl-3-(2-phenylethyl)piperidine
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(3-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
[(3R,4R)-1-[3-(dimethylamino)benzoyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
ethyl 4-{[4-(3-phenylprop-2-ynoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
4-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
N-ethyl-3-(4-methoxyphenyl)-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
5-{2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-cyclobutyl-7-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-methyl-1H-1,3-benzodiazol-5-yl]-2-methoxyacetamide
(4aR,7aS)-1-benzyl-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(thiophen-3-ylmethyl)acetamide
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]furan-2-carboxamide
N-[(3S,4R)-1-(5-acetylpyridin-2-yl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]propanamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4,4,4-trifluorobutan-1-one
4-(5,6-dimethylpyrimidin-4-yl)-N-[3-(4H-1,2,4-triazol-4-yl)phenyl]piperazine-1-carboxamide
N-{2-[7-(2-chloro-6-fluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-methylpropanamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
2-[1-(cyclohexylmethyl)-4-[4-(trifluoromethyl)pyrimidin-2-yl]piperazin-2-yl]ethan-1-ol
2-{2-[(3-methoxypyrrolidin-1-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
(5-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}furan-2-yl)methanol
methyl 3-[(2-chlorophenyl)methyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{1-[4-(4-fluorophenyl)butanoyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
3-(cycloheptylamino)-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
1-(naphthalene-1-carbonyl)-N-phenylpiperidin-3-amine
N-{1-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}methanesulfonamide
7-fluoro-2-methyl-3-{2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}-1H-indole
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(oxan-4-yl)ethyl]amine
(4aR,8aS)-1-butyl-6-[(3,4-difluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
3-{[2-amino-7-(3-methylbenzoyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}propan-1-ol
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(thiophen-3-yl)ethan-1-one
N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(5-oxo-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-methylpyrrolidine-2-carboxamide
N-[(2R,3R)-1'-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-(2-benzylmorpholin-4-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
(3S,4S)-1-(7-fluoro-2-methylquinoline-4-carbonyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
N-ethyl-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
4,6-dimethyl-1-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydropyrimidin-2-one
(2S)-2-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}amino)propanamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-4-(thiophen-2-yl)butan-1-one
N-cyclooctyl-2-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)acetamide
2-(1H-imidazol-1-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
2-[(3,5-difluorophenyl)methyl]-8-(1-methylcyclopropanecarbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-5-ethyl-1-methyl-1H-1,2,4-triazol-3-amine
N-(1-{7-cyclohexanecarbonyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-(dimethylamino)acetamide
6-(2-chlorophenyl)-N-(2-oxopiperidin-3-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(4-benzylpiperazine-1-carbonyl)-2-ethyl-6-methyl-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridin-4-one
(3aS,6aS)-2-methanesulfonyl-5-[2-(pyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(oxan-2-yl)ethyl]propanamide