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3-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]-N-methylbenzamide
N-({7-[(2-hydroxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methoxybenzamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-1-[4-(3-methoxyphenyl)piperazin-1-yl]propan-1-one
1-cyclopropyl-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
(4S)-4-(propan-2-yl)-3-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,3-oxazolidin-2-one
(3E)-4-phenyl-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]but-3-enoic acid
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(methylsulfanyl)propanamide
9-(4,6-dimethylpyridine-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-4-(3-methyl-3-phenylpiperidine-1-carbonyl)-1,3-thiazol-2-amine
2-(2-methoxyethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)acetamide
3-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-1-(cyclohex-1-en-1-ylmethyl)urea
6-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-1,3-benzothiazole
5-methyl-4-({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)thieno[2,3-d]pyrimidine-6-carboxylic acid
1-[5-methoxy-2-(2-methyl-1H-imidazol-4-yl)phenyl]-3,5-dimethyl-1H-pyrazole
2-(4-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}piperidin-1-yl)acetamide
6-ethyl-2-(3-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N,N-diethyl-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-(furan-2-ylmethyl)-2-methyl-N-(pyridin-2-ylmethyl)-5-sulfamoylbenzamide
1-[(2,3-dimethoxyphenyl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
3-[(3R,4S)-1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
5-(4-ethylpiperazine-1-carbonyl)-2-(3-fluorophenyl)-1,3-benzoxazole
2-(4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
1-[(4aR,8aR)-4a-hydroxy-7-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
4-[(3-methoxyphenyl)methyl]-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]piperazin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[N-(3-methylphenyl)methanesulfonamido]acetamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(1-phenylethyl)-1,2-oxazole-5-carboxamide
6-(difluoromethyl)-2-(3-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
8-(1-hydroxypropan-2-yl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-cyclopropyl-N-[(3-fluorophenyl)methyl]-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
3,7-dimethyl-11-({4-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-3,7,11-triazaspiro[5.6]dodecane
1-(2,5-dimethylfuran-3-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-(2-chlorophenyl)-1-(3-methoxypropyl)-3-{2-oxo-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
(1S,2S,3R,4R)-3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]bicyclo[2.2.1]heptan-2-amine
N-[(3,4-dimethoxyphenyl)methyl]-3,4-difluoro-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1,2-oxazole-5-carboxamide
N-methyl-N-[2-(piperidin-1-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(thiophen-2-yl)urea
N-(1,3-benzothiazol-2-ylmethyl)-2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methylacetamide
3-methyl-7-(pyridin-4-ylmethyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
{[3-({1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(furan-3-ylmethyl)methylamine
(1H-imidazol-2-ylmethyl)(methyl){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
1-{2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
(1S,5R)-6-(cyclobutylmethyl)-3-(4-methoxy-3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-fluorophenyl)-N-[1-(pyridin-2-yl)propyl]piperidin-4-amine
ethyl 2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
(2S)-1-[1-(6-fluoro-4-methylquinazolin-2-yl)piperidine-4-carbonyl]pyrrolidine-2-carboxamide
5-{1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]piperidin-4-yl}-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione