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N-[(2R,3R)-1'-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
2-[2-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1H-pyrrol-1-yl]pyrimidine
1-[3-(3-chlorobenzoyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-{[8-(2-phenylethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
4-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(4-methoxyphenyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-methyl-4-(1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
(4aS,7aR)-1-[(3-chlorophenyl)methyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
3-[2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]propanamide
N-cyclopropyl-N-(1-{1-[(2,5-difluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)furan-2-carboxamide
1-(4-{[4-(7-fluoro-2-methylquinoline-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
1-(cyclopent-1-ene-1-carbonyl)-3-(2,5-difluorobenzoyl)piperidine
4-[4-(cyclohex-3-ene-1-carbonyl)piperazin-1-yl]quinazoline
6-fluoro-2-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)quinolin-4-ol
N-cyclopropyl-1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-3-(thiophene-2-carbonyl)piperidine
{1-[(4-{[4-(methylsulfanyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidin-2-yl}methanol
6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[3-(2-methoxyacetamido)phenyl]-4-(morpholin-4-yl)piperidine-1-carboxamide
N-[4-(methylsulfanyl)phenyl]-6-[2-(4-phenylphenyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(2-chloro-5-methylphenyl)-3-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}urea
2-{N-methyl-1-[3-(1H-pyrazol-1-yl)phenyl]formamido}-2-(thiophen-2-yl)acetic acid
3-(3,4-difluorophenyl)-5-(1-methoxypropan-2-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-2,4-dimethylpyrimidine-5-carboxamide
N-[1-(4-chlorophenyl)ethyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
methyl 3-(2-methylbutyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-2-methoxy-2-phenylacetamide
N-[1-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(piperazine-1-carbonyl)benzene-1-sulfonamide
3-[1-(4-methylphenyl)cyclopentyl]-5-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,2,4-oxadiazole
N-benzyl-3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carboxamide
2-methyl-5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-1,3-benzodiazole
3-(furan-2-ylmethyl)-5-[1-(4-methylbenzoyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-[(4-methylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
3-{1-[(3-carboxypropyl)carbamoyl]piperidin-3-yl}benzoic acid
N-(3,4-difluorophenyl)-1-(3,5-dimethylfuran-2-carbonyl)piperidin-3-amine
N-[(2R,3R)-2-hydroxy-1'-[3-(thiophen-2-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
2-[1-cyclopropyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)acetamide
3-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxypyridine-3-carboxamide
1-(2-{1-oxa-8-azaspiro[4.5]decan-8-yl}pyrimidin-4-yl)pyrrolidin-3-ol
N-[1-(4-{[(5-ethylpyridin-2-yl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]-2,4-dimethylbenzamide
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
7-(6-chloro-2H-chromene-3-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-(5-methylhex-5-en-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1-{[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(furan-3-carbonyl)piperidine
(2S,4R)-4-amino-1-{[2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl}-N-methylpyrrolidine-2-carboxamide
N,N-dimethyl-2-(3-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carboxamide
1-[3-oxo-3-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one