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1-{1-[(3-methoxyphenyl)methyl]-5-(3-methylbut-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
1-{4-[(3-chloro-4-propoxyphenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
(3R,4S)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-propylpyrrolidin-3-amine
N-(adamantan-2-yl)-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
N-cyclopropyl-1-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)piperidine-4-carboxamide
6-(2,5-dimethylphenyl)-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[4-({cyclopropyl[(4-ethoxyphenyl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
4-[2-({5-methyl-4-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-yl]pyrimidin-2-yl}sulfanyl)ethyl]morpholine
5-(1-cyclobutanecarbonylpiperidin-4-yl)-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
1-{2-[2-(2H-1,3-benzodioxol-5-yl)acetamido]ethyl}-N-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
N-ethyl-2-(4-fluorophenyl)-N-(pyridin-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
5-(2-chlorophenyl)-N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]furan-2-carboxamide
2-fluoro-N-{3-[4-methyl-3-oxo-2-(propan-2-yl)piperazin-1-yl]-3-oxopropyl}benzamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
5-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
1-(4-cyano-2-ethylphenyl)-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
6-[(3-methoxyphenyl)methoxy]-4-(5-methylthiophene-2-carbonyl)-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
1-(furan-3-ylmethyl)-4-{[5-(methylsulfanyl)-4-phenyl-4H-1,2,4-triazol-3-yl]methyl}piperidine
6-phenyl-N-(1-phenylcyclopropyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-fluoro-2-{1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-2-yl}-1H-1,3-benzodiazole
1-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
3-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}benzonitrile
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-5,7-dimethyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
(2E)-N-{[7-(4-acetylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
1-(2-methylpropyl)-4-(3-phenyl-1,2-oxazole-5-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
4-[(2,3-dimethoxyphenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperazine-2-carboxylic acid
(2E)-3-(3-fluorophenyl)-1-(4-{3-[(4-phenylpiperazin-1-yl)methyl]phenoxy}piperidin-1-yl)prop-2-en-1-one
6-(5-methyl-1H-indol-3-yl)pyridin-2-amine
(1-{4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-3-methyl-1-oxobutan-2-yl)urea
1-(2-hydroxyethyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
1-(4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-[4-(dimethylamino)phenyl]-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl}ethan-1-ol
2-(3,5-dimethylfuran-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-({[7-methyl-2-oxo-1-(2-phenylethyl)-1,2-dihydroquinolin-3-yl]methyl}amino)-1λ6-thiolane-1,1-dione
1-(2-{3-cyclopropyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}ethyl)-5-methyl-1H-1,2,3,4-tetrazole
4-phenyl-N-[(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)methyl]benzamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
1-[(2E)-2-methylbut-2-en-1-yl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-cyclopropanecarbonyl-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidine-3-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]acetamide
1-[(3-methoxyphenyl)methyl]-4-(piperidin-4-yl)piperazin-2-one
4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]-1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidine
N-cyclohexyl-2-methyl-N-(pyridin-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-methyl-4-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,3-thiazol-2-amine
1-[2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)ethyl]piperidine-3-carboxamide
1-(pyridin-3-yl)-2-{4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazol-1-yl}ethan-1-ol