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3-methyl-5-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
3-(1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-1,3-oxazolidin-2-one
2-[3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1H-indol-1-yl]-N-(propan-2-yl)acetamide
1-(furan-2-carbonyl)-4-[3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperazine
1-(4-methoxyphenyl)-6,6-dimethyl-4-[2-(methylsulfanyl)benzoyl]piperazin-2-one
methyl 2-(1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
1-(2-methylphenyl)-4-(3-phenoxypropanoyl)piperazin-2-one
3-methyl-7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
6-fluoro-4-(2-methylpyrrolidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
1-cyclohexyl-4-[3-(pyridin-4-yl)propanoyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-(2-methylpropyl)-N-(oxolan-2-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
1-ethyl-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-methyl-4-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
7-(cyclobutylmethyl)-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-{[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-(pyridine-2-carbonyl)-1,4-diazepane
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-4-methylpiperazine-1-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-(3-hydroxy-2,2-dimethylpropyl)piperidine-3-carboxamide
3-butyl-1-methyl-4-{[(1s,4s)-4-aminocyclohexyl]methyl}piperazin-2-one
4-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}-1H-indole
[(3R,4R)-1-(2-ethoxybenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-[(4-chlorophenyl)methyl]-5-(3,4-dimethylpiperazine-1-carbonyl)-1,3-benzoxazole
N-[4-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)phenyl]acetamide
N-{2-[(2,6-dimethylphenyl)carbamoyl]phenyl}-4-(propan-2-yl)-1,2,3-thiadiazole-5-carboxamide
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[2-(methylsulfanyl)pyridine-3-carbonyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
(7S,9aR)-7-benzyl-N-(3-fluorophenyl)-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
6-methyl-2-{1-[2-(pyridin-2-yl)ethyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
3-(2-hydroxyphenyl)-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-1H-pyrazole-5-carboxamide
2-{2-[2-(methylsulfanyl)benzoyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
4-[4-oxo-7-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(pyridin-3-yl)propanamide
(1R,3S)-7-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-ol
6-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)pyrimidin-4-ol
(1S,5R)-6-propyl-3-{2-[2-(trifluoromethyl)phenyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-3-methoxypropanamide
2-[2-(dimethylamino)ethyl]-8-[3-(thiophen-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
N,N-dimethyl-3-[2-oxo-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanamide
1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
5-(azepane-1-carbonyl)-N-(cyclohexylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(3S,4S)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-propylpyrrolidine-3-carboxylic acid
2-(2-{1-[(2,6-dichlorophenyl)methyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
2-[4-(hydroxymethyl)phenyl]-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
N-[(3S,4R)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(3S,4S)-1-{[3-(methylsulfanyl)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
2-cyclopentyl-N-[3-(4-{[2-(3-methoxyphenyl)ethyl]amino}piperidin-1-yl)phenyl]acetamide