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(3S,4R)-4-(4-fluorophenyl)-1-{2-[4-(hydroxymethyl)phenyl]acetyl}pyrrolidine-3-carboxylic acid
N-[(2-fluorophenyl)methyl]-3-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]propanamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyridine
1-{1-[(3-methoxyphenyl)methyl]-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
2-{6-[(3-phenoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(pyridin-4-yl)ethan-1-one
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-2-(3-methoxyphenyl)azetidine
1-(4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
8-(7-chloro-1-methyl-1H-indole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[(4aS,8aR)-6-(9H-fluorene-9-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-5-methoxy-1H-indole-2-carboxamide
3-{2-oxo-2-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}-1,2,3-oxadiazol-3-ium-5-olate
(4aS,7aR)-1-[(2-methylpyrimidin-5-yl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-8-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-(3-methylpyridin-4-yl)-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1,4-diazepane
1-(4-fluoro-3-methoxybenzoyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
1,3-dimethyl-8-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3,5-dimethyl-1H-pyrrole-2-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[6-(1-hydroxyethyl)pyridin-2-yl]piperazin-2-one
2-(4-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}phenoxy)pyrimidine
N-[(2R,3R)-1'-[(3-fluorophenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxyacetamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(oxolan-2-ylmethyl)acetamide
3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-[(1-phenylcyclohexyl)methyl]propanamide
N-[2-(3-chlorophenyl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
1-[2-(4-methoxyphenyl)ethyl]-N3-methyl-N5-[(5-methylfuran-2-yl)methyl]-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-benzyl-4-hydroxypiperidine-1-sulfonamide
5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,7,8-trimethylquinoline-4-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(5-methylfuran-2-yl)ethyl]acetamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1-methylcyclopropanecarbonyl)piperidine
5-[3-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
3-(3-hydroxy-3-methylbutyl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
2-{1-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1H-1,2,3-triazol-4-yl}-1-ethyl-1H-1,3-benzodiazole
3-[(5-methyl-1,2-oxazol-3-yl)methyl]-1-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(2E)-3-phenylprop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-fluorophenyl)-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-one
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(4-methylphenoxy)acetamide
4-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}butanamide
N-(3-methoxypropyl)-6-[4-(piperidin-1-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-[5-benzyl-2-oxo-4-(1H-pyrazole-3-carbonyl)piperazin-1-yl]benzonitrile
(R)-cyclohexyl[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methanol
3-[5-(5-methylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-azabicyclo[2.2.2]octane
1-phenyl-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-[(1-ethylpiperidin-3-yl)methyl]-2-(1H-pyrazol-1-yl)benzamide
1-[3-({[(2-chlorophenyl)methyl]amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-3,6-diazabicyclo[3.2.2]nonane
1-{3-[4-(cycloheptylamino)piperidin-1-yl]phenyl}-3-methylimidazolidin-2-one
(3aS,6aR)-5-(4,6-dimethoxypyrimidin-2-yl)-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one