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1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[4-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]imidazolidin-2-one
2-(2-fluoro-3-methoxyphenyl)-1-methyl-1H-imidazole
1-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)urea
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-(oxan-4-ylmethyl)propanamide
4-cyano-1-methyl-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)-1H-pyrrole-2-carboxamide
2-butyl-6-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
N-[1-(2-chlorophenyl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-benzyl-N,1-dimethyl-5-{[2-(propan-2-yloxy)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 3-({4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}formamido)heptanoate
1-(pyridin-4-yl)-4-[(3R,5R)-5-(pyrrolidine-1-carbonyl)piperidine-3-carbonyl]piperazine
(1S,5R)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-4-acetamido-N-ethyl-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidine-2-carboxamide
N-(3-fluorophenyl)-N'-methyl-N'-[1-(pyridin-4-yl)ethyl]ethanediamide
(1S,5R)-3-methyl-6-{[2-methyl-5-(3-methyl-1H-pyrazol-5-yl)thiophen-3-yl]sulfonyl}-3,6-diazabicyclo[3.2.2]nonane
2-amino-N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-(quinolin-5-yl)pyrazin-2-amine
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(morpholin-4-yl)propyl]propanamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(2-methoxyethyl)-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxamide
2-[5-(methoxymethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-1,3-benzothiazole
(2E)-N-methyl-3-(pyridin-3-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]prop-2-enamide
N-(4-cyanonaphthalen-1-yl)-7-methyl-2,7-diazaspiro[4.4]nonane-2-carboxamide
2-[2-(dimethylamino)ethyl]-9-{[2-(propylamino)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)imidazo[1,2-a]pyridine-6-carboxamide
3-[(4-methoxyphenyl)methyl]-N-methyl-N-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
1-{[4-({1-[4-(piperidin-1-yl)benzoyl]piperidin-3-yl}methoxy)phenyl]methyl}-4-(pyridin-3-ylmethyl)piperazine
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-amine
(2E)-N-({7-[2-(4-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
(3R,4S)-1-(2-methyl-1,3-thiazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
ethyl 1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-2-carboxylate
2-[5-(3-chlorothiophen-2-yl)-1,2,4-oxadiazol-3-yl]pyrazine
N-(4-{[3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
{3-benzyl-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-yl}methanol
N-cyclohexyl-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-amido}piperidine-1-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(but-2-yn-1-yl)-5-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
6-fluoro-2-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
N-(2-methoxyethyl)-1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
methyl 8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
5-methyl-3-[2-(morpholin-4-yl)ethyl]-5-(1-{2-[3-(trifluoromethyl)phenyl]acetyl}piperidin-4-yl)imidazolidine-2,4-dione
N-[2-(dimethylamino)ethyl]-N-ethyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1,9-dimethyl-4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-tert-butyl-3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrrole
1-(4-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
3-cyclopropyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-5-carboxamide