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N-(cyclohexylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzamide
N-[4-(2-methoxypyridin-3-yl)-8-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-3-methylbutanamide
{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
N-[1-({[2-(1H-indol-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-phenoxyacetamide
N-ethyl-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxamide
N-[(1r,4r)-4-hydroxycyclohexyl]-1-benzofuran-3-carboxamide
4-({3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1H-indole
(2S)-2-(3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-3-phenylpropanamide
4-[4-(4-{[cyclohexyl(methyl)amino]methyl}-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyrimidin-2-amine
(2S,4R)-N,N-dimethyl-4-[(4-methylpyrimidin-2-yl)sulfanyl]-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
N-{[7-(5-fluoro-1H-indole-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-(2-methylphenyl)-3-(oxolan-3-yl)-5-(1H-pyrrol-3-yl)-1H-1,2,4-triazole
N-[3-(5-cyano-6-methoxy-2,4-dimethylpyridin-3-yl)phenyl]acetamide
3-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)benzonitrile
(3R,4S)-4-cyclopropyl-1-(7-methoxy-4-methylquinolin-2-yl)pyrrolidin-3-amine
2-[2-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
2,2-diethyl-4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]morpholine
N-{3-[1-(2,4-dimethylphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]propyl}acetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}thiophen-3-yl)methyl]dimethylamine
methyl 2-[3-methyl-2-oxo-4-(2-phenylpyrimidine-5-carbonyl)piperazin-1-yl]acetate
5-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
9-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-1-[1-(benzenesulfonyl)cyclopropanecarbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[4-(4-phenyl-1H-imidazol-1-yl)phenoxy]propanamide
1-ethyl-N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
N-cyclopropyl-1-{1-[(2,5-difluorophenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[2-(2,4-difluorophenyl)-1-[1-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]ethyl]-N-methylpropanamide
2-{5-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-1,3-benzodiazole
ethyl 1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
6-{[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroquinolin-2-one
ethyl 2-{[3-({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}carbamoyl)phenyl]amino}acetate
8-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-2-[4-(morpholin-4-yl)-2-(piperidin-1-yl)pyrimidin-5-yl]propanoic acid
9-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
methyl 2-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)sulfonyl]benzoate
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-phenoxypropan-1-one
(2S,4R)-4-amino-N,N-diethyl-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidine-2-carboxamide
N-[(2R,3R)-2-methoxy-1'-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
2-[2-(morpholin-4-ylmethyl)-4-(pyrazin-2-yl)phenoxy]-1-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}ethan-1-one
1-cyclohexyl-2-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
6-({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)-2-methylheptan-2-ol
1-(2-fluorophenyl)-N-[2-(pyridin-3-yloxy)propyl]cyclopropane-1-carboxamide
N-[(3S,4R)-1-[(6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
6-[1-(5-methoxy-3-methyl-1H-indole-2-carbonyl)piperidin-4-yl]pyrimidin-4-ol
N-{3-[({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}carbamoyl)methoxy]phenyl}propanamide
5-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]-1H-indole
5,5-dimethyl-3-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,3-oxazolidine-2,4-dione
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]benzamide