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2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide
4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
(1S,5R)-6-(cyclobutylmethyl)-3-[(3-hydroxy-4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(4-chlorophenyl)-N-[2-hydroxy-1-(thian-4-yl)ethyl]butanamide
N,N-dimethyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(2-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-1,3-thiazol-4-yl)methanol
1-[3-({6-[2-(2-hydroxyethyl)piperidine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-yl}amino)propyl]pyrrolidin-2-one
3-[5-({[2-(pyrrolidin-1-yl)ethyl]sulfanyl}methyl)-1,2,4-oxadiazol-3-yl]pyridazine
1-ethyl-8-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
[1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)piperidin-2-yl]methanol
N-{[5-(4-fluorophenyl)-1,2-oxazol-3-yl]methyl}-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(isoquinoline-3-carbonyl)-6-methoxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
methyl 3-(3-{2-[(4-methylphenyl)formamido]ethyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl)benzoate
N-benzyl-N,1-dimethyl-5-[4-(4-methylphenyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-5-{[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}furan-2-carboxamide
2-cyclopropyl-5-{4-[(4-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrimidin-4-ol
2-(cyclopropylmethyl)-8-[2-(1H-imidazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl (2S)-2-{[1-(6-methoxy-4-methylquinazolin-2-yl)pyrrolidin-2-yl]formamido}-3-methylbutanoate
5-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridin-2-amine
N-[1-(4-chlorophenyl)cyclobutyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
4-[(2-hydroxyethyl)sulfamoyl]-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-[2-(1H-imidazol-2-yl)benzoyl]piperidine
4-(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-amido)oxane-4-carboxylic acid
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-{[4-(methylsulfanyl)phenyl]methyl}cyclopropanamine
[(3R,4S)-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-(furan-2-yl)-1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]azepane
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(5-chloro-1H-1,3-benzodiazol-2-yl)acetamide
4-(4-acetamido-1H-pyrazol-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}benzamide
ethyl 1-({3-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperidine-4-carboxylate
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[(2S,4S)-2-{[(dimethylsulfamoyl)amino]methyl}-4-fluoropyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N,N-dimethyl-3-(1-{[3-(pyridin-2-yl)phenyl]methyl}piperidin-3-yl)propanamide
N-[3-({[2-(dimethylamino)-1-phenylethyl](methyl)carbamoyl}amino)-4-fluorophenyl]propanamide
ethyl 1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-[({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amino]propan-1-ol
1-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)-3-methylpentane-1,2-dione
5-acetamido-2-ethyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
4-[2-(2-methoxyphenyl)acetyl]-1-(2-methylphenyl)piperazin-2-one
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(2-methylphenyl)methyl]acetamide
2-amino-4-(furan-2-yl)-5-propyl-6-(pyridin-3-yl)pyridine-3-carbonitrile
ethyl 1-methyl-5-(1,2,5-thiadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]isoquinoline
(2R,6S)-2,6-dimethyl-4-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-4-yl)morpholine
3-[(1R,2S)-2-hydroxycyclohexyl]-3-methyl-1-[4-(thiophen-2-ylmethoxy)phenyl]urea
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
({5-[1-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine