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1-(6-cyclopropylpyrimidin-4-yl)-4-(pyridin-3-yl)piperidin-4-ol
(2S,4R)-N-(2,3-difluorophenyl)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
N-({1-[(6-chloroquinolin-2-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-(2-methyl-1H-imidazol-1-yl)butanamide
5-(5-fluoro-4-methoxypyrimidin-2-yl)-8-methoxyquinoline
ethyl 3-[(3-methoxyphenyl)methyl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine-3-carboxylate
3-(thiophen-3-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
3-(8-methoxy-2-methylquinolin-5-yl)-N,N-dimethyl-1H-1,2,4-triazol-5-amine
methyl 2-[4-(4-methoxyphenoxy)piperidin-1-yl]pyridine-3-carboxylate
2-(5-acetylthiophen-3-yl)-N-{2-[bis(propan-2-yl)amino]ethyl}acetamide
N-({7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
N-[(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-3-(pyridin-3-yl)propanamide
N-(cyclohexylmethyl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[5-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-1,2,4-oxadiazol-3-yl]benzoic acid
N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
methyl 8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-cyclohexyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1,3-benzoxazole-6-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-cyclopropanecarbonyl-8-{thieno[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[benzyl({7-chloro-4-[(oxolan-2-ylmethyl)amino]quinazolin-2-yl}methyl)amino]ethan-1-ol
3-(2-fluorophenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
5-[2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-imidazol-1-yl]-1-methylpiperidin-2-one
6-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)quinoline-4-carboxamide
4-propyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
7-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-N-(5-methylpyridin-3-yl)benzamide
2-(methylsulfanyl)-N-{[8-(pyridin-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
(2S,4R)-4-amino-N-methyl-1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]pyrrolidine-2-carboxamide
dimethyl(2-{[(3-methyl-1H-pyrazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}ethyl)amine
4-{3-[(E)-2-cyclohexylethenyl]-1-methyl-1H-1,2,4-triazol-5-yl}morpholine
4-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(pyrimidin-4-yl)ethyl]amine
4-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-2-phenylpyrimidine
ethyl 1-(1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperidine-3-carboxylate
N-[(2-chlorophenyl)methyl]-3-[1-(pyridin-4-yl)piperidin-3-yl]propanamide
1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-hydroxypropan-1-one
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(4-methoxy-2-methylbenzoyl)piperidine
N-cyclopropyl-2-[4-(1-methoxyethyl)phenyl]benzamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxybenzoyl)piperazine
3-methyl-N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
5-cyclopropyl-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-oxazole-4-carboxamide
2-(2-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-4-methyl-6-(trifluoromethyl)pyrimidine
4-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1,4-oxazepane
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-methyl-1-[(5-phenyl-1,2-oxazol-3-yl)methyl]urea
N-[(2R,3R)-2-ethoxy-1'-{[4-(2-hydroxyethoxy)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-{5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}-2-methylbutanamide
(2S,4S)-4-amino-N-ethyl-1-[2-(1H-1,2,4-triazol-3-ylsulfanyl)acetyl]pyrrolidine-2-carboxamide
4-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}piperazin-2-one
N-methyl-N-[2-(methylamino)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide