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N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyrrolidin-1-yl)acetamide
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
N-[(1S)-2-hydroxy-1-phenylethyl]-3-(4-hydroxyphenyl)benzamide
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}cyclopentanamine
9-[(2R,3S)-2-amino-3-hydroxybutanoyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(1,3-thiazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
3-{[2-(ethylsulfanyl)ethyl]carbamoyl}-5-methoxybenzoic acid
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(4-methylquinolin-2-yl)pyrrolidin-3-yl]acetamide
1-methyl-5-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
3-({[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}methyl)-1-(cyclohexylmethyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,6-dimethyl-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-benzyl-6-{[4-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
5-(2-methyl-1,3-thiazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-4-phenylbutanamide
2,3,5-trimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-ethyl-4-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
1-(2-fluorophenyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]cyclopropane-1-carboxamide
N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{1-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
1-[3-(3-methylpiperazine-1-carbonyl)benzenesulfonyl]azocane
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-indole-5-carboxamide
3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
1-methyl-8-(oxan-4-yl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-chloro-2-(furan-2-yl)-N-{2-[(2R)-pyrrolidin-2-yl]ethyl}quinoline-4-carboxamide
2-phenyl-1-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-yl)ethan-1-ol
(3aR,6aS)-5-[(2-ethoxyphenyl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-N-[1-(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]piperidine-4-carboxamide
3-[(3,3-difluoropyrrolidin-1-yl)methyl]-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
2-[2-(8-methoxy-2-methylquinolin-5-yl)phenoxy]propanamide
1-methyl-4-({6-[3-(propan-2-yloxy)phenyl]pyridin-3-yl}methyl)piperazine
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methylpropanamide
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-3,4-dimethoxypyridine
3-{1-[5-(1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methyl-4H-1,2,4-triazole
4-{4-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl]phenyl}-2-methylbutan-2-ol
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
(2S,4S)-4-amino-N-methyl-1-{[4-(2-methylpropyl)phenyl]methyl}pyrrolidine-2-carboxamide
2-(dimethylamino)-N-{3-methyl-1-[7-(naphthalene-1-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
[2-(1H-1,3-benzodiazol-2-yl)ethyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-[(2R,3R,6R)-5-(4-methoxy-3-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-[5-(1H-1,3-benzodiazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-methylpiperidin-2-one
3-(4-methoxyphenyl)-1-(3-methylbutyl)-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
(1S,5R)-6-(3,4-difluorobenzoyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(1,3-thiazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(2,5-dimethoxyphenyl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]ethan-1-one
N-[1-(1H-pyrazol-1-yl)propan-2-yl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide