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(4aS,7aR)-1-(4-chlorobenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,8aR)-1-(3-hydroxypropyl)-6-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-(oxan-2-ylmethyl)propanamide
1-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(cyclopropylmethyl)piperazine
N-benzyl-N-(1,3-thiazol-2-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
3-(1-{2-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(cyclobutylmethyl)-2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-(pyridin-3-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
8-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-oxa-8-azaspiro[4.6]undecane
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N,4-dimethyl-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[4-(methylsulfanyl)phenyl]propanamide
9-[(2,5-dimethylphenyl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[3-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
5-{1-[2-(4-chlorophenyl)acetyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
ethyl 4-(oxan-2-ylmethyl)-1-{[4-(trifluoromethyl)phenyl]carbamoyl}piperidine-4-carboxylate
(4aS,8aS)-4a-hydroxy-7-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-(propan-2-yl)-decahydro-2,7-naphthyridine-2-carboxamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propan-1-one
3-[(3R,4S)-1-(4-aminopyrimidin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-[2-(3-chloro-1-benzothiophen-2-yl)-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
N-[(4-fluorophenyl)methyl]-3-{1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}propanamide
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(quinolin-5-ylmethyl)acetamide
1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
1-(2,4-dimethylphenyl)-4-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]piperazine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(1R,7S)-6-(3-hydroxyazetidine-1-carbonyl)-3-[(5-methylpyrazin-2-yl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-(4-acetylbenzoyl)-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[1-(2-cyclohexylacetyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
methyl 1-(benzyloxy)-8-[(4-ethylphenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(2-{[(5-methyl-1,2-oxazol-3-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
5-[(3-fluorophenyl)methyl]-5-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)imidazolidine-2,4-dione
2-{1-[(4-ethoxyphenyl)methyl]-4-[(6-fluoroquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-(2H-1,3-benzodioxol-5-yl)-5-[(1S,2R)-2-(pyrrolidine-1-carbonyl)cyclohexyl]-1H-1,2,4-triazole
methyl 3-[(2-fluoro-4-methoxyphenyl)methyl]-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[1-(3,4-difluorophenyl)-5-(ethoxymethyl)-1H-1,2,4-triazol-3-yl]acetamide
6-[(2-fluorophenyl)methoxy]-4-(furan-2-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
4-[(3-methoxypropyl)amino]-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-(4-ethoxyphenyl)-3-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropanamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,4-difluorobenzamide
(2R,3R,6R)-5-(1-benzofuran-2-ylmethyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{[3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-oxazol-5-yl]methoxy}isoquinoline
(1R,3S)-3-[(2-phenylethyl)(pyridin-2-ylmethyl)carbamoyl]cyclopentane-1-carboxylic acid
N-({8-[(9-ethyl-9H-carbazol-3-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methylpropanamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
5-chloro-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]thiophene-2-carboxamide
(3S,9aR)-8-(4-methoxybenzoyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[1-(3-methylpyridin-2-yl)propan-2-yl]amine