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N-[4-({4-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepan-1-yl}methyl)phenyl]acetamide
7-(1-benzothiophen-3-yl)-4-(pyrrolidine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(1-methylpiperidin-4-yl)-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
5-(2,6-dimethylphenoxymethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
[2-(1H-indol-1-yl)ethyl](methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
7-(2-methoxyethyl)-2-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[4-(dimethyl-1,2-oxazol-4-yl)-6-methylpyrimidin-2-yl]phenol
3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-methyl-N-(pyridin-3-ylmethyl)aniline
2-[(1-methylpiperidin-2-yl)methyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(2-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
3-{2-[4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-4-[(3-methoxyphenyl)methyl]piperazin-2-one
6-(4-methylazepan-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-1-[4-(pentyloxy)phenyl]urea
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-3-phenoxypropan-1-one
{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl}methanol
(3aS,6aS)-2-[(1-ethyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[2-(1H-pyrazol-1-yl)ethyl]-1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperidine
(2S)-2-amino-3-(4-methoxyphenyl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]propan-1-one
N-(2-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}quinolin-5-yl)acetamide
2-({2-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-2-(pyridin-3-yl)ethan-1-ol
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-methoxy-4-[4-(thian-4-yl)piperazine-1-carbonyl]quinoline
1-cyclopentyl-N-[1-(furan-2-yl)ethyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
7-(1-benzothiophen-3-yl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-(pyridin-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(1-methylpiperidin-4-yl)piperidine
2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
3-[(4-{5-[(cyclohexylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
N-{3-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-3-oxopropyl}methanesulfonamide
3-{[cyclopropyl(pyridin-3-ylmethyl)amino]methyl}-6-methoxy-1,2-dihydroquinolin-2-one
3-(1-{[4-(hydroxymethyl)phenyl]methyl}-4-phenyl-1H-imidazol-5-yl)benzonitrile
6-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,2-dihydropyridin-2-one
2-(2,5-dioxoimidazolidin-4-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]acetamide
N-methyl-1-(2-phenylethyl)-N-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-amine
1-[1-(cyclopropanesulfonyl)piperidin-3-yl]-3-phenylpropan-1-one
1-(4-methoxyphenyl)-4-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butane-1,4-dione
3-(3-{2-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}phenyl)-1,3-oxazolidin-2-one
N-ethyl-6-methyl-5-[5-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
N-[(2R,3R)-1'-[(2,4-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
6-[(4-fluorophenyl)methoxy]-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-1-(propan-2-yl)-1,4-diazepan-2-one
N-[2-(2-fluorophenyl)-1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
8-[(2-ethoxyphenyl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[(5-ethylpyridin-2-yl)methyl]methylamine
N-(2-methoxyethyl)-1-methyl-2-oxo-N-(thiophen-3-ylmethyl)-1,2-dihydroquinoline-3-carboxamide
1-{5-[3-(2,5-difluorobenzoyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
ethyl 3-[(3-methoxyphenyl)methyl]-1-{[4-(2-oxoimidazolidin-1-yl)phenyl]methyl}piperidine-3-carboxylate
N-(2-aminoethyl)-2-methyl-4-phenylpyridine-3-carboxamide
3-({1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-4H-chromen-4-one
ethyl 1-(2,5-dimethylphenyl)-5-({[(4-sulfamoylphenyl)methyl]amino}methyl)-1H-pyrazole-4-carboxylate
4-fluoro-3-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}benzene-1-sulfonamide