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N-(cyclopropylmethyl)-2-[3-(4-methoxyphenyl)-1-(3-methylbutyl)-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
methyl 2-hydroxy-5-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)benzoate
1-(4-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]benzamide
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(1r,4r)-4-hydroxycyclohexyl]benzamide
3-{2-[4-(2,3-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
N-{[1-(isoquinolin-5-ylmethyl)piperidin-4-yl]methyl}-3-methylbut-2-enamide
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-4-carboxamide
4-{[2-(thiophen-2-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}morpholine
2-{1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-(prop-2-en-1-yloxy)benzamide
2,6-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]quinoline-4-carboxamide
2-({4-phenyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1H-imidazol-1-yl}methyl)pyridine
3-chloro-5-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
ethyl 4-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}piperazine-1-carboxylate
1-{2-[(6-methoxypyrimidin-4-yl)(methyl)amino]ethyl}piperidin-2-one
4-[(5-chlorothiophen-2-yl)methyl]-N-(pyridin-3-yl)morpholine-2-carboxamide
1-[4-(propan-2-yl)phenyl]-3-[3-(1H-1,2,4-triazol-1-yl)propyl]urea
1-(5-chloropyridin-2-yl)-4-[2-(methylsulfanyl)pyridine-3-carbonyl]piperazine
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
2-[(furan-2-ylmethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amino]butan-1-ol
7-fluoro-N-(isoquinolin-5-ylmethyl)-N,3-dimethyl-1H-indole-2-carboxamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl){[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
1-cyclobutanecarbonyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
1-(4-methoxybenzoyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
2-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-(propan-2-yl)-1H-imidazole
(2S,4R)-4-amino-N-methyl-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidine-2-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
7-(2,6-dimethylhept-5-en-1-yl)-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(3,5-dimethylphenyl)-3-{1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-oxopropanamide
methyl 2-(3-methylphenyl)-2-(pyridin-3-ylformamido)acetate
4-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-1-methylpiperazine-2-carboxylic acid
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methylpropanamide
3-methyl-6-[5-(pyridin-3-ylmethyl)-1,2,4-oxadiazol-3-yl]pyridazine
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methyl-1H-pyrrole-2-carboxamide
3-(6-methoxynaphthalene-2-carbonyl)-1-(oxan-4-yl)piperidine
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(pyrrolidin-1-yl)piperidin-3-yl]-N-[3-(morpholin-4-yl)propyl]propanamide
(2H-1,3-benzodioxol-5-ylmethyl)[2-(2,6-dimethoxyphenoxy)ethyl]amine
8-[(2-phenylphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-(cyclopropylmethyl)-8-(3-propyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-5,6,7,8-tetrahydroquinazolin-2-amine
2-(dimethylamino)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2-(3-methylphenyl)acetamide
1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}azetidin-3-ol
5-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-propylpyrimidin-2-amine
1-(2-{[cyclopropyl(ethyl)amino]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
N-methyl-2-(3,4,5-trifluorophenyl)pyridine-4-carboxamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-4-(quinolin-5-ylmethyl)-1,4-diazepan-2-one
4-(2-methoxyphenyl)-1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperidine
methyl 1-ethyl-3-(oxolane-3-amido)-5-[(2-phenylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate