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3-[3-(1H-pyrazol-5-yl)phenyl]pyridine
3-(diphenylmethyl)-5-(oxolan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-{[benzyl(methyl)amino]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
2-ethyl-4-methyl-5-{1-[1-(thiophen-3-yl)propan-2-yl]-1H-imidazol-2-yl}-1H-imidazole
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(2-methoxyethyl)-N-(propan-2-yl)propanamide
2-[4-carbamoyl-4-(piperidin-1-yl)piperidin-1-yl]-2-(3-fluoro-5-methylphenyl)acetic acid
[(3R,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-ethoxy-6-({[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}methyl)phenol
4,5-dimethyl-3-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2,3-dihydro-1,3-oxazol-2-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-6-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxamide
[(2-fluoro-4,5-dimethoxyphenyl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-2-ol
4-{2-[2-(2-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]ethyl}morpholine
1-methanesulfonyl-3-[4-(methylsulfanyl)benzoyl]piperidine
2-(azepan-1-yl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]acetamide
(1S,6R)-9-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
1-methyl-N-[2-(pyrazin-2-yl)ethyl]azepane-2-carboxamide
2-(dimethylamino)-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-(4-methylphenyl)acetamide
3-{imidazo[1,2-a]pyridine-2-carbonyl}-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N,2,8-trimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
(3S,4R)-1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
2-(2-ethylpyridine-4-carbonyl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
6-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-[(3R,4S)-1-(3-cyano-4,5,6-trimethylpyridin-2-yl)-4-cyclopropylpyrrolidin-3-yl]-2-methoxyacetamide
N-[2-(4-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]-2-methoxyacetamide
(3-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-oxopropyl)urea
N-({3-methyl-7-[2-(piperidin-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
1-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S)-2-{[1-(4-benzenesulfonamidophenyl)piperidin-4-yl]amino}-3-phenylpropanamide
2-(benzylsulfanyl)-5-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyrimidine
1,3-dimethyl-4-{2-methyl-3-[(pyridin-3-ylmethyl)amino]benzoyl}piperazin-2-one
1-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}piperidin-3-ol
(4aS,7aR)-1-(1H-indole-5-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 2-[2-({4-[4-(oxolane-3-amido)-1H-pyrazol-1-yl]phenyl}formamido)ethyl]-1,3-thiazole-4-carboxylate
N-[1-(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]pyridine-3-carboxamide
8-[(5-methylfuran-2-yl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-hydroxypiperidin-1-yl)acetamide
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]pyrazine-2-carboxamide
2-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
1-methyl-4-(6-phenylpyridazin-3-yl)piperazine-2-carboxylic acid
3-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
6-(4-benzylpiperidine-1-carbonyl)-5-methyl-N-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(6-methylpyridin-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(1R,2R)-N-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-2-phenylcyclopropane-1-carboxamide
2-(furan-2-amido)-7-oxo-N-[3-(propan-2-yloxy)propyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
(3S,4S)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(propan-2-yloxy)pyrrolidin-3-ol