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5-({[(3-{2-[4-(2-chlorobenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
2-[5-(2,3-dihydro-1,4-benzodioxin-2-yl)-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
1'-benzoyl-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-ethyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,2,5-trimethyl-1H-pyrrole-3-carboxamide
N-[(2,4-difluorophenyl)methyl]-4-propylpyrimidine-5-carboxamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(pyridin-2-ylmethyl)propanamide
2-{5-[(2,4-dioxoimidazolidin-1-yl)methyl]-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
1-{4-[(2,3-difluoro-6-methoxyphenyl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
5-cyclopropyl-N-(2-methoxyethyl)-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
N-methyl-2-(3-methylbenzamido)-7-oxo-N-(1,3-thiazol-2-ylmethyl)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-benzyl-8-cyclohexyl-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-2-amine
1-{1-[6-(aminomethyl)-2-methylpyrimidin-4-yl]piperidin-4-yl}-2-phenylethan-1-ol
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-chloro-4-methoxybenzoyl)azepan-4-amine
(1R,5R)-N,N-dimethyl-6-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-[(4aR,7aS)-4-cyclohexanecarbonyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
6-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(2-ethyl-1,3-dihydroxypropan-2-yl)-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-N-cyclohexylbenzene-1-sulfonamide
2-{4-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
1-ethyl-3-[3-(3-methoxypropyl)piperidin-1-yl]piperidine
ethyl 2-{1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-amido]cyclohexyl}acetate
methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(3-phenylbutyl)amine
5-(3-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-oxopropyl)-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
6-methyl-3-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[2-(pyridin-3-yloxy)acetyl]-1,4-diazepan-5-one
3-chloro-N-(2-methoxyethyl)-4-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)benzamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
N-[(2,4-dihydroxyphenyl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-oxopentanamide
3-(pyrazin-2-yl)-1-(7-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-(4-acetylphenoxy)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methanesulfonyl-2-methylpyrimidin-4-amine
2-[4-(3,4-dimethylpiperazine-1-carbonyl)piperidin-1-yl]-4-methyl-6-(propan-2-yl)quinazoline
8-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)sulfonyl]-2,8-diazaspiro[4.5]decan-3-one
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(2-methoxyphenyl)methyl]amine
5-[5-(2-chlorophenyl)furan-2-carbonyl]-N-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
3-[(2,3-dihydro-1H-inden-2-yl)amino]-2-(thiophen-2-ylmethyl)propan-1-ol
2-ethyl-N-[(3-methyl-1-benzofuran-2-yl)methyl]pyrimidine-5-carboxamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-2-yl)ethyl]acetamide
3-[3-(1H-imidazol-2-yl)propyl]-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
7-(2-ethoxypyridine-3-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
6-oxo-N-[(1r,4r)-4-hydroxycyclohexyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide