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{7-fluoro-5-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
methyl 2-[(4-fluorophenyl)sulfamoyl]-6-[3-(methylsulfanyl)propyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(dimethylamino)-2-(4-methylphenyl)-1-[3-(piperidin-1-yl)azetidin-1-yl]ethan-1-one
(1r,4r)-4-({[5-(oxolan-2-yl)thiophen-2-yl]formamido}methyl)cyclohexane-1-carboxylic acid
N,1,3-trimethyl-N-[(3-methyl-1H-indol-2-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(6-hydroxy-6-methylheptan-2-yl)acetamide
3-(2-oxoimidazolidin-1-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)benzamide
4-(5-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)piperazin-2-one
N-{1-[7-(3,4-dimethylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}pyridine-2-carboxamide
3-(methoxymethyl)-1-{3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methylbenzoyl)piperidine
(1R,5S,6S)-6-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
4-({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)-1-phenylpiperazin-2-one
5-{[2-(dimethylamino)ethyl]carbamoyl}-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxylic acid
methyl 2-{[2-(3-fluorophenyl)ethyl]sulfamoyl}-6-[(2E)-2-methylbut-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-propyl-2-{4-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]morpholin-3-yl}acetamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[2-(2-methyl-1H-indol-3-yl)ethyl]amine
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-{spiro[indene-1,4'-piperidine]-1'-yl}propan-1-one
2-{3-[2-(azepane-1-carbonyl)morpholine-4-carbonyl]-5-methyl-1H-pyrazol-1-yl}-N-methylacetamide
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-4-(5-methylfuran-2-yl)benzamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3-methylphenyl)ethan-1-one
7-(cyclopropylmethyl)-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-ethylmorpholin-2-yl)ethyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
8-[3-(dimethylamino)propanoyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
[5-(1-benzothiophen-2-ylmethyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
3-[(4-methanesulfonamidopiperidin-1-yl)methyl]-N-(pyridin-4-yl)benzamide
2-oxo-4-[(E)-2-phenylethenyl]-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
N-(2-hydroxyethyl)-3-[5-(5-methoxyfuran-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
1-(3-methylbut-2-en-1-yl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-cyclohexyl-1-[1,3-dioxo-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
N4-[1-(furan-2-carbonyl)piperidin-3-yl]-6-(morpholin-4-yl)pyrimidine-2,4-diamine
1-{imidazo[1,2-b]pyridazin-6-yl}-4-[(4-methanesulfonylphenyl)methyl]piperazine
2-(2-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyridine
N-butyl-N-methyl-3-({[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)azepan-4-yl]thiophene-2-carboxamide
1-(2-cyclohexylethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(2-amino-4-{[2-(1H-imidazol-4-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-3-methylbut-2-en-1-one
6-(4-ethylphenyl)-N-(2-methylprop-2-en-1-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(diphenylmethyl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1,2-oxazole-5-carboxamide
5-({methyl[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
(4aS,8aR)-6-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-1-butyl-decahydro-1,6-naphthyridin-2-one
4-(4-butanoylpiperazin-1-yl)-2-[(2,3-dimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
4-[(4-methylphenyl)methyl]-3-{2-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
1-benzyl-3-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)urea
3-benzyl-8-[(3,5-difluorophenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N2-cyclopropyl-N4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(3S,4R)-1-{2-[methyl(1-methylpiperidin-4-yl)amino]acetyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid