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N-(1-{7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
5-methoxy-2-({3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(4-chloro-2-methylbenzoyl)piperidine
4-(3-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}propoxy)benzamide
1-[7-(3-chlorophenyl)-9-(pyridin-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
2-methyl-9-[2-(oxan-2-ylmethoxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
9-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-3-oxa-9-azaspiro[5.5]undecane
3-(2-chlorophenyl)-3-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)pyrrolidine-2,5-dione
[(2S,6S)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
6-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
7-cyclohexyl-2-[4-(dimethylamino)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
5-methanesulfonyl-2-methyl-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrimidin-4-amine
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methyl-6-(propan-2-yl)pyrimidine
5-{1-[2-(3,4-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-(3-chloro-4-fluorophenyl)-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}propanamide
2-{1-cyclohexyl-4-[6-(trifluoromethyl)pyridin-2-yl]piperazin-2-yl}ethan-1-ol
1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-(1H-pyrazol-1-yl)propan-1-one
2-methyl-1-[1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
2-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)phenoxy]-1-(pyrrolidin-1-yl)ethan-1-one
4-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)morpholine
(2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(1H-pyrrole-2-carbonyl)pyrrolidine-2-carboxamide
(3aR,6aS)-1-oxo-5-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-ethyl-5-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}pyrimidine
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
2-[benzyl(methyl)amino]-N-[2-(pyridin-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3,3-dimethylbutan-1-one
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-3-phenylprop-2-yn-1-one
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-4-cyclopropyl-1-[2-(2-ethoxyphenyl)acetyl]pyrrolidine-3-carboxylic acid
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
N-[4-(4-{[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]-5-phenylpentanamide
N-({3-methyl-7-[2-(2,3,6-trifluorophenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-2-methyl-N-[2-(piperidin-1-yl)ethyl]-1H-pyrrole-3-carboxamide
2-butyl-6-methyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyrimidin-4-amine
(2E)-3-(2-chlorophenyl)-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)prop-2-enamide
2-[4-(hydroxymethyl)phenyl]-1-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
N,1-dimethyl-3-(2-methylpropyl)-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
ethyl 4-(oxan-2-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(2R,3S,6R)-5-(4-chloro-1H-pyrazole-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4,7-dimethylquinazolin-2-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
4-[(dimethylamino)methyl]-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}azepan-4-ol
8-fluoro-3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
2-(2-methoxyethyl)-9-[(1-propyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methylprop-2-en-1-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-[(4-{6-[ethyl(methyl)amino]pyrimidin-4-yl}piperazin-1-yl)methyl]benzoic acid
5-benzenesulfonamido-1-ethyl-N-[(3-fluorophenyl)methyl]-2-methyl-1H-1,3-benzodiazole-7-carboxamide
N-cyclopropyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[3-(oxan-2-ylmethoxy)phenyl]methyl}benzamide
N3-[3-(4-chlorophenyl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide