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2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-[3-(propan-2-yloxy)benzoyl]piperidine
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
2-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-4-(pyridin-4-yl)pyrimidine
1-cyclopropyl-4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrrolidin-2-one
N-(isoquinolin-5-ylmethyl)-N,1-dimethyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
2-[2-(2,3-dimethylphenoxy)ethyl]-4-methoxypyrimidine
N-benzyl-2-[1-ethyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}acetamide
1-[1-(3-cyclopropylpropanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-cyano-N-(2,3-dihydro-1H-inden-2-yl)-N-methylbenzamide
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-3,6-dimethyl-2-(1-propyl-1H-pyrazol-4-yl)quinoline
(3aR,6aR)-2-(dimethylsulfamoyl)-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[6-(dimethylamino)pyrimidin-4-yl]benzamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
(3S,5R)-N3-butyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-(1H-1,3-benzodiazol-2-ylmethoxy)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
3-benzyl-8-[(5-chloro-2-hydroxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2E)-3-(2-chlorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]prop-2-en-1-one
5-{1-[(3-methyl-1-benzofuran-2-yl)methyl]-1H-1,2,3-triazol-4-yl}pyrimidine
(3R,4S)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-phenylpyrrolidin-3-amine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(isoquinoline-1-carbonyl)piperidin-3-amine
2-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
1-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decane
4-(3,6-dimethylpyrazin-2-yl)-2-[(2-ethylpiperidin-1-yl)methyl]phenol
1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
6-oxo-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-(5-methylfuran-2-yl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-5-carboxamide
3-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-1-[(5-ethylpyridin-2-yl)methyl]-1-methylurea
3-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
N,N,4-trimethyl-3-({[1-methyl-1-(methylcarbamoyl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
1-phenyl-N-[2-(propane-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]cyclopropane-1-carboxamide
3-[5-(1-methyl-1H-imidazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]benzonitrile
1-methyl-N-[2-(morpholin-4-yl)ethyl]-5-phenyl-1H-pyrrole-2-carboxamide
2-(4-chloro-2-methylphenoxy)-1-[3-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-3-ene-1-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-[4-(methylsulfanyl)phenyl]acetamide
4-[2-(4-fluorophenyl)piperidine-1-carbonyl]pyridazine
(3S,4S)-4-(dimethylamino)-1-[3-(piperidine-1-carbonyl)benzenesulfonyl]pyrrolidin-3-ol
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyridine-4-carboxamide
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
4-ethyl-1-methyl-3-{1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-chloro-5-(8-methoxyquinolin-5-yl)-N-methylbenzamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-methyl-N-[2-(methylamino)ethyl]piperidine-3-carboxamide
7-(2-methoxyethyl)-2-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide