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ethyl 3-[(3-methoxyphenyl)methyl]-1-(pyridine-3-carbonyl)piperidine-3-carboxylate
(7R,9aR)-N-benzyl-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-tert-butyl-3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[2-amino-4-(4-methoxyphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)(1,3-thiazol-4-ylmethyl)amine
3-methyl-5-[2-(3-methyl-3-phenylpiperidin-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}methyl)-N-ethylpyrimidin-2-amine
1-ethyl-5-[(oxan-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-{1-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-2-(2-phenylethyl)piperidine
3-[(2,5-dimethoxyphenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(3-methoxybenzoyl)piperidine
ethyl 1-(3-{[(1-hydroxycyclohexyl)methyl]carbamoyl}-6-[4-(methylsulfanyl)phenyl]pyridin-2-yl)piperidine-4-carboxylate
2-[4-(1-methylpiperidine-2-carbonyl)piperazin-1-yl]benzonitrile
2-(4-methoxyphenyl)-N-methyl-N-(oxan-2-ylmethyl)acetamide
1-[1-(cyclohex-1-en-1-yl)ethyl]-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)urea
N-[2-(4-methoxyphenyl)ethyl]-2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}acetamide
2-(4-chloro-2-{[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl}phenoxy)acetamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(oxan-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(2R)-pyrrolidine-2-carbonyl]piperidine
N-[(3S,4R)-4-(propan-2-yl)-1-{2-[4-(trifluoromethyl)phenyl]acetyl}pyrrolidin-3-yl]acetamide
1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]urea
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-4-methyl-1,2,5-oxadiazole-3-carboxamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-methoxyphenyl)methyl]propanamide
1-(5-{[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
4-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-5-(4-fluorophenyl)-2-methylpyrimidine
2-chloro-N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-fluorobenzamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{1-oxaspiro[4.4]nonan-3-yl}acetamide
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})[1-(pyrazin-2-yl)propan-2-yl]amine
4-[(5-acetylthiophen-3-yl)methyl]-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
2-[4-(2,3-dihydro-1H-inden-2-yl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
1-butyl-5-(2-{[(3-methylphenyl)methyl]amino}ethyl)pyrrolidin-2-one
N-[3-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)phenyl]-2-methylfuran-3-carboxamide
2-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]-6-ethoxy-4-methylquinazoline
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
[benzyl(methyl)sulfamoyl][(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]amine
1-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N-methyl-5-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}pyrimidin-2-amine
2-(5-methyl-1,2-oxazol-3-yl)-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)piperidine-1-carboxamide
5-cyclopropyl-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,3,4-oxadiazol-2-amine
5-ethyl-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(1-{4-[(2,3-dihydro-1H-inden-1-yl)carbamoyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
1-{5-[(1R,5S)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
N,2,3,6-tetramethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-{2-oxo-2-[4-(2-phenylethyl)piperidin-1-yl]ethyl}-4-(pyridin-3-ylmethyl)piperazin-2-one
2-(2-oxo-4-{[4-(2-phenylethoxy)phenyl]methyl}piperazin-1-yl)acetic acid