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N-[(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
1-[4-(2-amino-6-methylpyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-3-methylbut-2-en-1-one
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-4-carboxamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-ethyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}benzamide
4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-1-phenylpiperazin-2-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
3-(2-methoxyphenyl)-N-[1-({[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
2-(azepan-1-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}acetamide
methyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
2-[2-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
(3S,9aR)-3-benzyl-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(morpholin-4-yl)ethan-1-one
(3S,4S)-1-(benzenesulfonyl)-4-{methyl[2-(oxan-4-yl)ethyl]amino}pyrrolidin-3-ol
ethyl 4-{6-methyl-3-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]quinolin-2-yl}piperazine-1-carboxylate
8-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[({1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-4-yl}oxy)methyl]pyridine
N-methyl-N-[2-(2,3,6-trimethylphenoxy)ethyl]azepane-4-carboxamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl){[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
3-{[2-(2-fluoro-5-methoxyphenyl)-1H-imidazol-1-yl]methyl}-N-methylbenzamide
[3-(furan-2-ylmethyl)-9-[(5-methylthiophen-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4-(2-methylquinolin-6-yl)piperidin-4-ol
3-{2-oxo-2-[3-oxo-4-(2-phenylphenyl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
(3aS,6aS)-2-[(3-hydroxy-4-methoxyphenyl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-4-(propan-2-yloxy)benzamide
N-[(4-fluorophenyl)methyl]-2-(2-methoxyphenoxy)-N-(prop-2-en-1-yl)propanamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(4-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-cyclopentyl-1-{4-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}ethan-1-one
1-[(2-chloro-5-fluorophenyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-benzyl-3-(2-methoxyethyl)-8-[(2,3,4-trimethoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-5-methyl-2-phenyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazole-4-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
1-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-[4-(methylsulfanyl)phenyl]ethan-1-one
[(3-{[1-(2,3-dimethoxybenzoyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(1,3-thiazol-4-ylmethyl)amine
N-[2-(3-chlorophenyl)ethyl]-2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-6-(2-methoxyphenyl)pyridine-3-carboxamide
4-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane-1-carbaldehyde
ethyl 5-(furan-2-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(4-{[4-(2-ethylpiperidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazin-1-yl)pyrimidine
3-{2-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1-cyclopropyl-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
1-[6-hydroxy-4-(1H-imidazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
3-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-5-(dimethylsulfamoyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]benzamide
1-(1H-pyrazole-3-carbonyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
8-[(3-chloro-4-fluorophenyl)methyl]-3-[2-(dimethylamino)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-methoxy-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanamido]phenyl}-3-methylbutanamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one