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6-(benzyloxy)-4-[2-(1H-imidazol-2-yl)benzoyl]-1-(oxan-4-ylmethyl)-1,4-diazepan-2-one
2-[(1S,5R)-3-(1H-indole-6-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
{1-[2-({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-yl}methanol
2-(morpholin-4-yl)-1-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}propan-1-one
N-[(2R,3R)-2-methoxy-1'-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
methyl(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
6-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
[(3R,5R)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]propan-1-one
N-benzyl-N-methyl-3-({[2-(pyridin-3-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
3-[4-fluoro-3-(hydroxymethyl)phenyl]-4-methoxybenzamide
1-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-4-(pyridin-2-ylmethyl)piperazine
1-(4-{[1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methoxy}phenyl)-1H-1,2,3,4-tetrazole
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)propanamide
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
3-{2-[4-(2,4-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
4-(5-methoxypyridin-3-yl)-6-(1H-pyrazol-1-yl)pyrimidine
N-(propan-2-yl)-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
1-[(2-chloro-4-fluorophenyl)methyl]-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-1H-imidazole-2-carboxamide
N-({4-hydroxy-1-[2-(pyridin-3-yl)acetyl]azepan-4-yl}methyl)-2,5-dimethylfuran-3-carboxamide
1-ethyl-N-(3-methoxypropyl)-3,5-dimethyl-N-[(4-methylphenyl)methyl]-1H-pyrazole-4-carboxamide
3-({2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)benzoic acid
N-[1-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
methyl 3-[4-(2-methylpropyl)benzoyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-methyl-6-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
{1-[1-(naphthalen-1-ylmethyl)piperidin-3-yl]piperidin-4-yl}methanol
1-(2-methoxyethyl)-4-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]pyrrolidin-2-one
1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperazine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
4-{3-[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]propyl}morpholine
3-(1-methyl-1H-pyrazol-4-yl)-1-[2-(2-phenylethyl)morpholin-4-yl]propan-1-one
(3R,4R)-4-ethyl-1-{[4-(morpholine-4-sulfonyl)phenyl]methyl}piperidine-3,4-diol
methyl 6-(2-{[2-(3,4-difluorophenyl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(pyrrolidine-1-sulfonyl)amino]acetic acid
6-[(4-benzylpiperidin-1-yl)methyl]-2-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
5-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
5-(2-methoxy-4-methylphenoxymethyl)-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-oxazole-3-carboxamide
2-{2-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]phenoxy}ethan-1-ol
3-{2-[1-(butan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrrol-1-yl}pyridine
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
3-(1-acetylpiperidin-4-yl)-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(4-fluorophenyl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-methyl-1H-pyrazole-5-carboxamide
ethyl 1-[(4-methoxyphenyl)methyl]-5-[2-(pyrimidin-2-ylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[(E)-2-(4-hydroxy-3-methoxyphenyl)ethenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N,N-dimethyl-4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(methoxymethyl)piperidine
1-methyl-3-propyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide