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1-(3-{2-[(benzylamino)methyl]-4-methoxyphenoxy}-2-hydroxypropyl)piperidin-4-ol
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
N-{[8-(4-fluorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-4-(propan-2-yloxy)benzamide
1-[1-(4-methanesulfonylphenyl)ethyl]-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
3-{[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]sulfamoyl}-N-(prop-2-en-1-yl)benzamide
(1S,5R)-6-(3-chlorobenzoyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
7-(1,3-benzothiazol-2-yl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]methyl}benzoic acid
1-{[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-3-(4-methylphenyl)propan-1-ol
(4S)-4-(propan-2-yl)-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3-oxazolidin-2-one
2-{2-[2-(4-fluorophenyl)azetidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
1-methyl-9-[(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)methyl]-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
3-[(4-methoxyphenyl)methyl]-5-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazole
2-amino-6-(2-fluoropyridin-4-yl)pyrimidin-4-ol
4-acetamido-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}benzamide
2-[(2H-1,3-benzodioxol-5-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
S-[2-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-hydroxybutane-1-sulfonamido
2-(but-3-enoyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5,6-dimethyl-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(2-methylphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
methyl 4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}benzoate
N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
N-{[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
5-methyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-(1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
(3S,7S)-5-cyclopentanecarbonyl-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-benzyl-N-(2-hydroxyethyl)-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
1-methyl-4-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1,4,9-triazaspiro[5.5]undecane
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
3-[3-(propan-2-yloxy)benzoyl]-1-(1,3-thiazole-5-carbonyl)piperidine
4-methyl-N-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1,3-oxazole-5-carboxamide
N,N-dimethyl-3-{1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}propanamide
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-N-[(5-methylfuran-2-yl)methyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
4-methoxy-3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}benzene-1-sulfonamide
2-[(4-chlorophenyl)methyl]-8-(morpholine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-(1H-imidazol-1-ylmethyl)-1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-4-ol
2-(3-hydroxyphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
1-[1-ethyl-5-(3-methylthiophene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
1-[4-(quinazolin-4-yl)piperazin-1-yl]-4-(thiophen-2-yl)butan-1-one
4-[2-(methylsulfanyl)phenyl]-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-1-ethylpyrrolidin-2-one
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}oxan-4-amine
4-ethyl-1-methyl-3-({1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-ethyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrimidine-5-carboxamide
4-methyl-2-[1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-cyclopentanecarbonylpiperidine-4-carboxamide
4-({4-[(1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperidin-3-yl)methoxy]phenyl}methyl)morpholine
3-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-N-[1-methyl-3-(methylsulfanyl)-1H-1,2,4-triazol-5-yl]benzamide
2-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(2,2-dimethylpropyl)piperazin-2-yl)ethan-1-ol