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N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-1-ethyl-6-oxopiperidine-3-carboxamide
2-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]pyridin-3-ol
2-(4-ethylbenzenesulfonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-(3-methoxypropyl)-1-methyl-N-[(1-methyl-1H-indol-6-yl)methyl]piperidin-4-amine
(2R,6R)-4-[(2-carboxyphenyl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(4-methoxyphenyl)methyl]-3-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
2-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
4-(4-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}phenyl)-2-methylbutan-2-ol
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidin-4-ol
2-[2-hydroxy-2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N,N,3-trimethyl-4-({[2-(2-methylpropanesulfonyl)ethyl]carbamoyl}amino)benzamide
1-[(5-methylfuran-2-yl)methyl]-N3-[(3-methylphenyl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
4-(2-benzyl-1,3-benzoxazole-5-carbonyl)-1-cyclopentylpiperazin-2-one
N-cyclopropyl-1-[(1s,4s)-4-(4-phenylbenzenesulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-{2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
5-[(dimethylsulfamoyl)amino]-1-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-(3-methoxyphenyl)pyrrolidin-3-yl]-2-cyclopentylacetamide
1-(2-methylpropyl)-4-(2-phenoxyacetyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-(4-fluorophenoxymethyl)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
N-[1-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(butylsulfanyl)-N4-[2-(1,3-thiazol-4-yl)ethyl]pyrimidine-4,6-diamine
1-[(2-fluorophenyl)methyl]-5-(thiomorpholine-4-carbonyl)piperidin-2-one
5-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(4aR,7aS)-1-cyclobutanecarbonyl-4-(5-methyl-1,3-oxazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2-methoxyphenyl)methyl]-N-[2-(methylsulfanyl)ethyl]-6-oxopiperidine-3-carboxamide
(2S)-N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-(methylamino)propanamide
1-cyclohexyl-4-cyclopentyl-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
methyl 3-butanoyl-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3aR,7aS)-2-{[5-(1,2-oxazol-5-yl)thiophen-2-yl]sulfonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(3S,4S)-4-cyclopropyl-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
N-ethyl-3-(propan-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-5-carboxamide
2-{4-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
4-ethyl-3-[(1-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}piperidin-4-yl)methyl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,8aS)-2-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-decahydroisoquinolin-4a-ol
1-[(4-fluorophenyl)methyl]-4-[2-(2-methoxyphenoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
N-{[7-(dimethyl-1,3-thiazole-5-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2,6-difluorobenzamide
N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-2-(trifluoromethyl)benzamide
3-{[bis(pyridin-3-ylmethyl)amino]methyl}pyrrolidin-3-ol
(3R,9aR)-8-(3-methylbutyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(1H-imidazol-1-yl)propyl]-3-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-5-(phenylsulfamoyl)benzamide
2-methoxy-1-[1'-(quinoxalin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
{1-[4-(4-{[(3-chlorophenyl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
(2R,6S)-2,6-dimethyl-4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}morpholine
5-[5-(5-propyl-1,2-oxazol-3-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
1-[(4-fluorophenyl)methyl]-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(naphthalen-1-ylmethyl)acetamide