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4-({ethyl[(4-ethylphenyl)methyl]amino}methyl)-N-methylbenzene-1-sulfonamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-oxo-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
8-(1-ethyl-1H-pyrazole-5-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[6-(thiomorpholin-4-yl)pyridazin-3-yl]benzoic acid
2-(4-methyl-1H-pyrazol-1-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)acetamide
N-[2-(dimethylsulfamoyl)ethyl]-3-(4-hydroxyphenyl)-2-phenylpropanamide
7-(2-methylphenyl)-4-(pyrimidin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2,5-dimethoxyphenyl)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
N-({7-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
4-{3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-methyl-6-(1H-pyrazol-1-yl)pyrimidine
6-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
1-methyl-3-{1-[(1-methylpiperidin-4-yl)methyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-butyl-4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-4-(4-methoxyphenyl)-4-oxobutanamide
1-{1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]piperidin-4-yl}piperidin-4-ol
2-[4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]pyrimidine
2-methoxy-1-(4-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1,4-diazepan-1-yl)ethan-1-one
3-(azepane-1-carbonyl)-1-methyl-N-[(6-methylpyridin-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[1-(7-chloro-9-oxo-9H-fluorene-1-carbonyl)piperidin-4-yl]-N-cyclopropylpropanamide
(3aR,6aR)-2-acetyl-5-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
6-methoxy-1-[(4-methoxyphenyl)methyl]-4-[2-(3,4,5-trimethoxyphenyl)acetyl]-1,4-diazepan-2-one
3-({1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}oxy)pyridine
(3aR,6aR)-2-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(3,4-dimethoxyphenyl)methyl]-N-methylacetamide
2-methyl-5-[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]pyrazine
N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N3-cyclooctyl-N5-[1-(furan-2-yl)ethyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(4aR,8aS)-1-(3-ethoxypropyl)-6-[(2-hydroxynaphthalen-1-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-{1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}piperidin-4-ol
N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]carbamoyl}methoxy)phenyl]propanamide
N-{1-[(4-hydroxy-6-methylquinolin-2-yl)methyl]pyrrolidin-3-yl}acetamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-(2,5-dimethoxyphenyl)-2-(thiomorpholin-4-yl)acetic acid
1-(3-methoxyphenyl)-4-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazin-2-one
1-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}urea
(5S,9aS,9bS)-5-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(1-{2-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
14-[4-(1H-imidazol-1-yl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-ethyl-2-{4-[(3-fluoropyridin-2-yl)methyl]piperazin-1-yl}acetamide
N-[2-(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)ethyl]acetamide
2-(2-phenyl-1,3-thiazol-4-yl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
6-(benzyloxy)-1-cyclohexyl-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,4-diazepan-2-one
methyl 1-[(3R,5S)-1-(1-propylpiperidin-4-yl)-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
[2-(1-benzylpyrrolidin-3-yl)ethyl]({[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl})amine
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-4-methyl-2-phenylpyrimidine-5-carboxamide
1-(2-{1-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-[(3-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3R,7S,8aS)-7-{[(2,4-difluorophenyl)methyl]amino}-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione