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(1-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
3-ethyl-4-[(4-{[(4-methylphenyl)methyl]amino}quinazolin-2-yl)methyl]piperazin-2-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-cyclopropyl-6-oxo-N-[(4-phenyloxan-4-yl)methyl]piperidine-3-carboxamide
1-[4-({[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]imidazolidin-2-one
4-{3-[3-(2-hydroxyethyl)-4-methylpiperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-ethoxy-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
7-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-({3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
1-(2-methoxyethyl)-8-(3-phenylpropyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
methyl 3-[(3S,4R)-1-[(3,5-dimethoxyphenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propanoate
2-methoxy-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
5-methoxy-1-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1H-indole-2-carboxamide
5-benzamido-1-cyclopentyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-[2-(benzylsulfanyl)ethyl]-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(2-methoxyphenoxy)-N-{[8-(thiophene-2-sulfonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
4-(4-chlorophenoxy)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methylpiperidine-4-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(pyrrolidin-1-yl)propanamide
3-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-6-phenylpyridazine
1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-1,4-diazepane-6-carboxylic acid
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
1-(2-{1-cyclohexyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-1,2-dihydropyridin-2-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
9-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N-benzyl-1-(2-cycloheptyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-ethylpiperidine-4-carboxamide
5-methanesulfonamido-N-methyl-N-[(4-methylphenyl)methyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
methyl 4-({1-[2-(4-chlorophenyl)ethyl]-6-oxopiperidin-3-yl}formamido)butanoate
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}pyrazin-2-amine
N-(2H-1,3-benzodioxol-5-yl)-1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
4-(2H-1,3-benzodioxol-5-yl)-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[benzyl(methyl)amino]-3-[4-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}benzoic acid
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylpiperidin-3-amine
2-cyclooctyl-4-{4-[2-(3,4-dimethoxyphenyl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[3-(pyridin-4-yl)propyl]pyrimidine-5-carboxamide
N-[1-(1H-imidazol-4-ylmethyl)azepan-4-yl]-4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-(1,3,7-trimethyl-1H-indole-2-carbonyl)piperidin-3-yl]propanoic acid
3-[2-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
4-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-(cyclopentylmethyl)-3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-1-(3-methoxypropyl)-6-methyl-1,4-dihydropyridin-4-one
N-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-1,2,5-thiadiazole-3-carboxamide
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]pyridin-3-ol
1-(oxan-4-yl)-4-(1,3-thiazol-2-ylmethyl)piperazine
methyl 6-[(2,4-difluorophenyl)methyl]-2-[(1-methoxypropan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-(cyclohex-3-en-1-ylmethyl)-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1H-pyrrole-2-carboxamide
3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
N,5,6-trimethyl-2-oxo-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1,2-dihydropyridine-3-carboxamide