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N-{[4-(aminomethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-(2-{7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
N-(5-fluoro-2-methylphenyl)-2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)acetamide
[3-propyl-1-(pyrimidin-5-ylmethyl)piperidin-3-yl]methanol
1-[2-(dimethylamino)-4-{[1-(3-methylpyridin-2-yl)propan-2-yl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-(1-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)cyclopentan-1-ol
1-{1-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]ethyl}-4-methylpiperazine
[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)(1,3-thiazol-2-ylmethyl)amine
2-(3-hydroxyphenyl)-1-(4-methyl-3-phenylpiperazin-1-yl)ethan-1-one
N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-[(1R,3R)-3-aminocyclopentyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[4-(propan-2-yl)benzoyl]pyrrolidin-3-yl]methanol
3-[(3R,4S)-3-[2-(4-methylphenoxy)acetamido]-4-(propan-2-yl)pyrrolidin-1-yl]propanamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N-{[4-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperidin-4-ol
N-[(2R,3R)-2-methoxy-1'-[(3-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
1-cyclopropyl-3-(4-methoxyphenyl)-3-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
4-ethyl-5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
[3-(1H-imidazol-1-yl)propyl]({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})(pyridin-3-ylmethyl)amine
N-(5-methylpyridin-2-yl)-5-{1-[2-(1H-pyrazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-{[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]methyl}pyridine
1-(3-methoxyphenyl)-4-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperazin-2-one
4-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[4-(2-ethylbutyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-[(2R,3R)-1'-[(3,4-dimethylphenyl)methyl]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(oxolan-3-yl)-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-methyl-N-{2-[methyl(oxan-2-ylmethyl)carbamoyl]phenyl}furan-3-carboxamide
[(3R,4R)-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
methyl 3-[(2,4-dimethoxyphenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2-{2-[2-(dimethylamino)ethoxy]phenyl}phenyl)methanamine
N,6-dimethyl-N-(1,2-oxazol-3-ylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-[(2R,3R)-3-[benzyl(methyl)amino]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]propan-1-one
1-(2-{4-[(3-methoxypyrrolidin-1-yl)methyl]phenoxy}ethyl)-1H-imidazole
N-(3-hydroxy-3-phenylpropyl)-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(3-fluorophenyl)-3-[4-(piperidin-1-yl)piperidin-1-yl]-1,2,4-triazine
N-(1-benzothiophen-2-ylmethyl)-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
9-[2-(2,4-dimethylphenoxy)ethyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
8-[2-(2,4-dichlorophenoxy)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidin-4-amine
2-ethyl-4-({4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}methyl)pyrimidine
1-(2-cyclohexylethyl)-3-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
(4aR,8aS)-6-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
4-methyl-3-[({[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}carbamoyl)amino]benzamide
3-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-(4-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-amine
1-[1-(propan-2-yl)piperidine-4-carbonyl]-4-(4H-1,2,4-triazol-3-yl)piperidine