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3-(2-amino-1,3-thiazol-4-yl)-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)propanamide
2-[(3-methylpiperidin-1-yl)methyl]-4-(pyrimidin-2-yl)phenol
2-{4-[(4-chlorophenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-methyl-3-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1H-pyrazol-5-yl]-2-phenoxypropanamide
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-[(4-fluorophenyl)methyl]piperidine
ethyl 1-{[4-(methoxycarbonyl)phenyl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(quinolin-4-ylmethyl)-1,2-oxazole-3-carboxamide
6-[2-(cyclohex-1-en-1-yl)acetyl]-3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-[2-({4-[1-(furan-3-carbonyl)piperidin-3-yl]-5-methylpyrimidin-2-yl}sulfanyl)ethyl]morpholine
1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
N-[(3R,4S)-4-cyclopropyl-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
N-(3,5-dimethylphenyl)-6-(2,2-dimethylpropanoyl)-6-azaspiro[2.5]octane-1-carboxamide
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-1-(piperidin-1-yl)ethan-1-one
(5S,9aS,9bS)-5-(3-hydroxyphenyl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3R)-3-cyclopropyl-4,4-dimethyl-1-(1,3-thiazole-4-carbonyl)pyrrolidin-3-ol
2-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-N-(2-ethylphenyl)-2-oxoacetamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-{[3-methyl-7-(4-methyl-2-oxopentanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-indole-2-carboxamide
(3aR,6aR)-2-[3-(3-fluorophenyl)propanoyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 2-[1-(quinoxaline-6-carbonyl)piperidin-2-yl]acetate
(1S,5R)-3-{imidazo[1,2-a]pyridine-2-carbonyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N-diethyl-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-(pyridin-3-yl)piperidin-4-ol
1-cyclopentyl-N-methyl-6-oxo-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}piperidine-3-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]propanamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(4-ethylphenyl)methyl]-N-methylbenzamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
(1H-indol-4-ylmethyl)({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
3-[5-(9H-purin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(4-methoxyphenyl)methyl]piperidine
N-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
7-[(4-fluorophenyl)methyl]-2-(2-methylbenzoyl)-2,7-diazaspiro[4.5]decane
2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyrazine
3-(1-propyl-1H-1,3-benzodiazol-5-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
3-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-methylpropan-1-one
N-[2-(3-methoxyphenyl)ethyl]-4-(piperidin-3-yl)benzamide
propyl 2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
8-[(2,4-dimethylphenyl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[4-(furan-2-yl)phenyl]methyl}(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
methyl 4-({1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)butanoate
methyl 3-[(2-cyclopentylacetamido)methyl]-5-(quinoline-8-sulfonamido)benzoate
4-(4-acetylbenzoyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
methyl 4-{[4-benzyl-4-(hydroxymethyl)piperidine-1-carbonyl]amino}benzoate
(2S)-1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(methylamino)propan-1-one
3-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
methyl (2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-[methyl(pyridin-2-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
N-(propan-2-yl)-1-[(1s,4s)-4-{[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(3S,4R)-1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide