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(3S,5R)-N3-(6-methylpyridin-3-yl)-N5-[(3-methylthiophen-2-yl)methyl]piperidine-3,5-dicarboxamide
5-(propan-2-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclohexyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
2-[(1S,5R)-3-(6-aminopyrimidin-4-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
4-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1,3-thiazole-5-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[1-(propan-2-yl)piperidine-3-carbonyl]piperazine
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-3-{imidazo[1,2-a]pyridin-2-yl}-N-methylpropanamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidine-3-carboxylic acid
N-{[5-chloro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetamide
1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetamide
1-(2-phenylethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-ol
5-(4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxymethyl)furan-2-carboxylic acid
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}quinoline-6-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
{1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}methanol
5-{2-[(3-methoxyphenyl)amino]butanoyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-benzyl-N,5-dimethyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(quinolin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[4-(furan-2-yl)phenyl]methyl}-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
2-[1-(propan-2-yl)piperidin-4-yl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]acetamide
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-(pyridin-3-yl)ethane-1,2-dione
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(oxan-4-yl)acetamide
8-cyclopropanecarbonyl-2-[(4-fluorophenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetamide
1-[4-(morpholine-4-carbonyl)phenyl]-N-{[3-(trifluoromethoxy)phenyl]methyl}piperidin-4-amine
N-cyclobutyl-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
8-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(2S)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]pyrrolidine-2-carbonyl]morpholine
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)methylamine
2-[(3R,4R)-3-[(4-ethylpiperazin-1-yl)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-5,6-dimethylpyridine-3-carbonitrile
2-(2-{[2-(1H-indol-3-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-(4-fluorophenyl)-N-[(2S)-1-hydroxybutan-2-yl]quinoline-4-carboxamide
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(prop-2-en-1-ylsulfanyl)propan-1-one
N-[2-(3-methylpyridin-2-yl)ethyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
1-[(5-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}thiophen-2-yl)methyl]pyrrolidine
1-[3-(2-fluorophenoxy)azetidin-1-yl]-4-(piperidin-1-yl)butan-1-one
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-4-ylmethyl)piperazine
2-amino-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
N-(2-{[2-(dimethylamino)-2,3-dihydro-1H-inden-2-yl]formamido}ethyl)pyridine-3-carboxamide
2-{[(1R,2S)-2-phenylcyclopropyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-N'-(4-methylphenyl)propanediamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(hydroxymethyl)piperidin-4-ol