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ethyl 5-({[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]amino}methyl)furan-2-carboxylate
2-methyl-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-amino-6-(2,5-dimethylphenyl)-4-[5-(hydroxymethyl)furan-2-yl]pyridine-3-carbonitrile
3-[(1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-4-yl)oxy]pyridine
5-fluoro-2-(1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
10-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
3-[(2-methoxyphenyl)methyl]-5-[(1-methylpyrrolidin-2-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-[(4-ethylphenyl)methyl]-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-(4-methoxyphenyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
ethyl 4-[6-(cyclopent-1-ene-1-carbonyl)-6-azaspiro[2.5]octane-1-carbonyl]piperazine-1-carboxylate
1-(2-{[(5-methanesulfonyl-2-methylphenyl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
(1S,5R)-6-benzyl-3-[(5-methylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-cyclopentylpyrrolidine-3-carboxylic acid
4-(hydroxymethyl)-1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-ol
7-(furan-3-carbonyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl({[2-(morpholin-4-yl)quinolin-3-yl]methyl})[2-(pyridin-2-yl)ethyl]amine
3-[(4-fluorophenyl)formamido]-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
4-[1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-1,2,3-triazol-4-yl]benzonitrile
1-[(4-methyl-1H-imidazol-5-yl)methyl]-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methyl-N-(pyrimidin-4-ylmethyl)acetamide
8-chloro-2-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,3-triazole
N-(2-chloro-5-methylphenyl)-4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carboxamide
1-methyl-8-{[4-(methylsulfanyl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(2-chlorophenyl)-3-{1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-(dimethylamino)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-methylpyrimidine-5-carboxamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(oxolan-3-ylmethyl)acetamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]propanoic acid
1-{4-[2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
5-methyl-N-[(1R,2S)-2-phenylcyclopropyl]-1-propyl-1H-pyrazole-4-carboxamide
2-[3-(oxolan-3-yl)-5-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl]acetic acid
2-methoxyethyl N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylcarbamate
2-(3-methylbut-2-en-1-yl)-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
3-amino-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
3-(1H-indazol-5-yl)-1-[2-(3-methoxy-4-propoxyphenyl)ethyl]urea
3-(3-fluoro-4-phenylbenzoyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
5-(4-methyl-1H-pyrazol-1-yl)pyridine-3-carboxamide
2-(2-hydroxyphenyl)-1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
6-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}pyridine-2-carbonitrile
1,6-dimethyl-3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
(4aR,7aS)-1-cyclopropanecarbonyl-4-(3-methyl-1,2-oxazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
1-[(4aR,8aR)-7-[(3,4-dimethoxyphenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
4-(2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}ethyl)morpholine
2-methyl-3-{[3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}-1H-indole