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7-(2-hydroxyethyl)-2-(1H-1,2,3-triazol-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-{3-[(2-amino-6-methylpyrimidin-4-yl)amino]propyl}phenol
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[3-(propan-2-yloxy)propyl]-1H-1,3-benzodiazole-7-carboxamide
3-methyl-N-[(1-methylpiperidin-4-yl)methyl]-4-phenyl-1,2-oxazol-5-amine
methyl (2S,4R)-1-[(4-ethoxyphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
N,3,5,7-tetramethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-indole-2-carboxamide
3-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2S,4R,6S)-2-(2-methylpropyl)-6-[4-(pyridin-2-yl)phenyl]oxan-4-yl]acetamide
(2R)-N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]oxolane-2-carboxamide
N-methyl-5-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
1-methyl-3-propyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
1-[(3-fluorophenyl)methyl]-N-methyl-6-oxo-N-(quinolin-2-ylmethyl)piperidine-3-carboxamide
N-methyl-2-(phenylamino)-N-[1-(1,3-thiazol-5-yl)ethyl]pyrimidine-5-carboxamide
4-(3,3-diphenylpiperidine-1-carbonyl)-1-ethylpyrrolidin-2-one
5-{[4-(3,4-dichlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-methyl-1H-imidazole
2-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
(2R)-2-cyclohexyl-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxyethan-1-one
2-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-5-(4-hydroxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-(2-methylphenoxymethyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}piperidine
5-acetyl-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}thiophene-3-carboxamide
methyl 4-[5-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
3-[5-(cyclohex-3-en-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-cyclopropylpropanamide
(2E)-3-(3,4-dimethoxyphenyl)-1-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}prop-2-en-1-one
2-butyl-4-({2-[(2-methylpyrrolidin-1-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)-1H-imidazole
4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-3-(thiophen-2-yl)-1H-pyrazole
ethyl 2-{2-cyclopropanecarbonyl-2,7-diazaspiro[4.5]decan-7-yl}acetate
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methoxypyrimidine
4-[6-(methoxymethyl)pyrimidin-4-yl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-amino-8-hydroxy-4-[5-(hydroxymethyl)furan-2-yl]-5H,6H-benzo[h]quinoline-3-carbonitrile
N-[2-(dimethylamino)-1-phenylethyl]-N-methyl-5,6,7,8-tetrahydroquinoline-3-carboxamide
1-{4-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
N-[2-(dimethylamino)ethyl]-6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(hydroxymethyl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-ol
methyl({[5-(oxan-2-yl)furan-2-yl]methyl}){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-(oxan-3-yl)-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
1-[3-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-oxopropyl]-1,2-dihydropyridin-2-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-cyclopropyl-9-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-5-[4-(5-methyl-1H-indazole-3-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
1-(2-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]phenoxy}ethyl)-4-ethylpiperazine
5-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-N,N-dimethylpyridin-2-amine
{3-[(3-methoxyphenyl)methyl]-1-[3-(5-methylfuran-2-yl)benzoyl]piperidin-3-yl}methanol
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]pyridazine-3-carboxamide
5-[methyl(2-phenylethyl)amino]-2-[2-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)-2-oxoethyl]-2,3-dihydropyridazin-3-one
ethyl 2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)acetate
N-cyclobutyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
8-chloro-2-[1-(piperidin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]quinoline