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ethyl (4aS,8aR)-6-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylate
5-propyl-1'-(quinolin-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{2-[5-methyl-4-({methyl[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]amino}methyl)-1,3-oxazol-2-yl]phenyl}thiophene-3-carboxamide
3-[(4-cyclopentylpyrimidin-2-yl)amino]propanamide
N-[2-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxolane-2-carboxamide
3-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-N,N-dimethylaniline
(1S,5R)-3-benzyl-6-(2-ethylpyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}-1H-indole
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(oxan-4-yl)acetamide
2-{8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
7-[(2,3-difluorophenyl)methyl]-2-(3,3-dimethylbutanoyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(3-fluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-methyl-2-(piperidin-1-yl)pyrimidine-5-carboxamide
(3R,4R)-1-(1,3-benzoxazol-2-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
methyl 4-({1-ethyl-3-methyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)benzoate
(3S,4R)-N,N-dimethyl-1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]-4-propylpyrrolidin-3-amine
3-[3-(cyclopropylmethyl)-5-(pyrazin-2-yl)-1H-1,2,4-triazol-1-yl]-4-fluorobenzene-1-sulfonamide
(3S,9aR)-8-(3,5-dichlorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclopropyl-4-methoxy-2-({1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}oxy)benzamide
3-(2-methylpropyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-5-carboxamide
4-[4-(2,5-dimethylphenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-{3-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenyl}acetamide
2-amino-4-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-7-methyl-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
N-cyclohexyl-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)-N-methylpropanamide
3-[2-(azepan-1-yl)-2-oxoethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
1-{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}piperidine-4-carboxamide
(3S,4R)-1-(4-butylbenzoyl)-4-methylpiperidine-3,4-diol
(1S,2R)-N1-cyclopropyl-N1-[(3-ethoxyphenyl)methyl]-N2-methylcyclohexane-1,2-dicarboxamide
2-methyl-5-({3-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-1,3-benzothiazole
5-benzoyl-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-[(3,5-dimethoxyphenyl)methoxy]-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-(propan-2-yl)-1,4-diazepan-2-one
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
N4,N4,5-trimethyl-N2-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-2,4-diamine
(2S,4S)-4-amino-N-methyl-1-[(E)-2-phenylethenesulfonyl]pyrrolidine-2-carboxamide
1-[(5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-2-methoxyphenyl)methyl]-1H-1,2,4-triazole
N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]pyrrolidin-3-yl]methanol
3-[(2-fluorophenyl)formamido]-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[1-(pyrazin-2-yl)propan-2-yl]amine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-1H-1,3-benzodiazole-5-carboxamide
2-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-5-fluoro-3-methyl-1H-indole
5-(oxane-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-({3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-3,5-dimethyl-1H-pyrazole
1,5-dimethyl-2-phenyl-4-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
N-[(1-methylpyrrolidin-3-yl)methyl]-2-propoxybenzamide
2-(4-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}morpholin-2-yl)ethan-1-amine
3-benzyl-4-(dimethyl-1,2-oxazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4S)-N-(3-chloro-2-fluorophenyl)-3-hydroxy-4-(morpholin-4-yl)pyrrolidine-1-carboxamide