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2-ethyl-N-methyl-N-[1-(pyridin-3-yl)pentyl]pyrimidine-5-carboxamide
4-methyl-2-{1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
2-{4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
4-ethyl-3-[1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-benzamido-5-methylphenyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(pyridin-4-yl)piperazine
2-{[5-(1-methoxyethyl)-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
6-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]pyridine-2-carboxylic acid
({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
2-(2-{[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenoxy)ethan-1-ol
[1-(5-{[(4-fluoro-2-methoxyphenyl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
methyl (2S,4S)-1-[(3-methylphenyl)methyl]-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-N'-phenylethanediamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-(2-hydroxypropyl)-1,2-oxazole-3-carboxamide
ethyl 2-[(1R,5S,6S)-6-[(furan-3-ylmethyl)(methyl)carbamoyl]-3-azabicyclo[3.1.0]hexan-3-yl]acetate
N,N-diethyl-1-{1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-benzothiophene-5-carboxamide
6-[(2E)-2-methylbut-2-enoyl]-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
(2E)-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-3-(thiophen-2-yl)prop-2-enamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-1,1-dioxo-2,5-dihydro-1λ6-thiophene-3-sulfonamide
2-methyl-1-({3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
2-{1-[(4-ethoxyphenyl)methyl]-4-[6-methyl-2-(methylamino)pyrimidin-4-yl]piperazin-2-yl}ethan-1-ol
8-[3-(propan-2-yl)-5-[(pyrimidin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]quinoline
1-({3-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]phenyl}methyl)-1H-pyrazole
3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
methyl (2S,4R)-4-[3-(1H-1,2,3-benzotriazol-1-yl)propanamido]-1-methylpyrrolidine-2-carboxylate
6-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]quinoxaline
5-({[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3,5,7-trimethyl-1H-indole-2-carboxamide
3-methanesulfonamido-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
4-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}thiomorpholine
2-[1-(1-methylpiperidin-4-yl)-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-2-yl]ethan-1-ol
N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-(4-fluorophenyl)-4-[1-(3-methoxy-4-methylbenzoyl)piperidin-3-yl]piperazine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
(2S,6S)-1-(1H-imidazol-4-ylmethyl)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
(2S,4S)-4-amino-N-ethyl-1-{[2-(2-phenylethynyl)phenyl]methyl}pyrrolidine-2-carboxamide
2-{[4-(2-fluoro-5-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}benzonitrile
3-[2-(thiophen-2-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]phenol
3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-N,N-dimethylaniline
3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(propan-2-yloxy)pyridazine
(4aR,7aS)-1-{2-[4-(propan-2-yl)piperidin-1-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-(propan-2-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
4-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-2-(trifluoromethyl)morpholine
N,2,5-trimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-oxazole-4-carboxamide
N-{4-fluoro-3-[({[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}carbamoyl)amino]phenyl}acetamide
N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(3-{1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-yl}piperidin-1-yl)acetamide
2-{2-[3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
8-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one