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8-(6-cyclopropylpyrimidin-4-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[9-(3-methyl-1,2-oxazole-5-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
4-(1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)morpholine
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-ethyl-N-(oxan-2-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-2-(4-fluorophenyl)-N-(furan-2-ylmethyl)acetamide
4-cyano-N-(3-acetamido-4-methoxyphenyl)piperidine-1-carboxamide
N,N-dimethyl-7-(oxane-4-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3S,9aR)-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2S)-1-cyclohexyl-3-hydroxypropan-2-yl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-(5-phenyl-1H-pyrazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]pyridin-2-amine
N-butyl-N-(furan-2-ylmethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
5-ethyl-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine
5-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-2-methyl-1,4-dihydropyridin-4-one
1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
1-{3,4-dihydrospiro[1-benzopyran-2,1'-cyclopentane]-4-yl}-3-(1-ethyl-1H-pyrazol-5-yl)urea
N-{[4-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
N-(2-fluoro-5-methylphenyl)-3-[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]propanamide
1-(2-methylpyridin-4-yl)-4-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-1,4-diazepane
1-(4-cyclohexylpiperazin-1-yl)-2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]ethan-1-one
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxamide
1-[(2R,3R)-2-hydroxy-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(methylsulfanyl)ethan-1-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-phenyl-1H-pyrazole-4-carboxamide
1-(3-fluoro-2-methylphenyl)-3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}urea
N-[(3S,4R)-4-(4-methylphenyl)-1-[2-(phenylsulfanyl)ethyl]pyrrolidin-3-yl]acetamide
2-[5-(2,3-difluoro-6-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
2-ethyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
[1-(2-{[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}ethyl)piperidin-3-yl]methanol
3-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-cyclopropylpropanamide
N-{2-[(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)formamido]ethyl}pyridine-3-carboxamide
2-ethoxy-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)pyridine-3-carboxamide
3-(cyclopropylmethyl)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidine-3-carboxylic acid
N,5,7-trimethyl-N-[3-(oxolan-2-yl)propyl]pyrido[2,3-d]pyrimidin-4-amine
4-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperazine-2-carbonyl]morpholine
4-[4-(4-hydroxyphenyl)butan-2-yl]-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
N-[2-({[3-(3-methoxyphenyl)phenyl]carbamoyl}amino)ethyl]-2-methylpropanamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[2-(1H-indol-1-yl)ethyl]methylamine
(2S,4S,5R)-1,2-dimethyl-5-phenyl-4-[(pyridin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-3-methyl-1H-pyrazole-4-carboxamide
(3aR,6aS)-5-(3-fluoro-4-methoxybenzenesulfonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-ethyl-6-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
3-[2-(pyridin-3-yl)-1,3-benzoxazol-5-yl]propan-1-ol
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(2-hydroxyphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)piperidine-3-carboxamide
ethyl 9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxylate
3-(1-methyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
(8R,9aS)-8-hydroxy-2-[2-(quinolin-8-yloxy)ethyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
2-(3,4-dichlorophenyl)-4-[2-(pyridin-2-yl)ethyl]morpholine
3-(2-{1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}ethyl)phenol