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4-({1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-2-yl}methyl)morpholine
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(3S,4R)-1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
5-chloro-4,6-dimethyl-3-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]-1,2-dihydropyridin-2-one
N-(1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-[(5-methylfuran-2-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(2S)-2-{[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]amino}-4-(methylsulfanyl)butan-1-ol
(3aS,6aS)-N-(4-cyano-2-ethylphenyl)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrole-2-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[(2-methylphenyl)methyl]benzamide
9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-4-(pyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
3-methyl-7-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-fluoro-N-({1-[3-(thiophen-2-yl)propanoyl]piperidin-3-yl}methyl)benzamide
2-(adamantan-1-yl)-4-hydroxy-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
2-{4-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperazin-1-yl}phenol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-(pyridin-2-yl)pyrimidin-2-amine
N-benzyl-1-cyclopropyl-5-(3-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-(2-phenylpropyl)-1H-pyrazole-4-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-[(1-methylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-(methoxymethyl)-3-{[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
N-[2-(dimethylamino)ethyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
7-(cyclohexylmethyl)-2-(3-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(4-methylphenyl)methyl]amino}methyl)piperidin-2-one
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
(2S)-N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-amino-3-phenylpropanamide
N,1,3,6-tetramethyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
4-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}benzene-1-sulfonamide
2-ethyl-N-{3-[(2-ethylphenyl)carbamoyl]phenyl}pyrimidine-5-carboxamide
4,6-dimethyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-methoxy-N-({7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
7-methyl-2-(quinoline-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(1-{2-[(4-methylpyridin-2-yl)amino]ethyl}-4-phenyl-1H-imidazol-5-yl)benzonitrile
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-(2-methoxyethyl)-4-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
3-[3-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
3-(4-fluorophenyl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
1-(2-oxo-2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)pyrrolidin-2-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-(pyridin-3-ylmethyl)acetamide
9-[(3-fluoro-2-methylphenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-methoxy-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
4-(5-{1-[(5-methylfuran-2-yl)methyl]pyrrolidin-2-yl}thiophene-2-carbonyl)-1,4-oxazepane
ethyl 2-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-2-yl}acetate
2-ethyl-9-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(2-aminoethyl)-N-[2-(1H-indol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(4-ethylphenoxy)ethyl]-2-{imidazo[1,2-a]pyridin-3-yl}-N-methylacetamide