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2-(pyridin-2-ylmethyl)-9-[3-(pyridin-3-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylsulfamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-2-(2-fluorophenyl)acetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-(1H-pyrazol-1-yl)propanamide
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[2-(3-methoxyphenyl)ethyl]-N-{[4-(methylsulfanyl)phenyl]methyl}oxolane-3-carboxamide
[(5-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}thiophen-3-yl)methyl]dimethylamine
3-{2-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
(3S)-3-[4-(2,4,6-trimethoxyphenyl)-1H-1,2,3-triazol-1-yl]azepan-2-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]acetamide
2-(4-{[1-(1H-imidazol-1-yl)propan-2-yl]amino}piperidin-1-yl)pyridine-3-carbonitrile
4-(1H-imidazol-1-ylmethyl)-1-[3-(methylsulfanyl)propyl]piperidine
N-cyclopentyl-2-[cyclopropyl(1H-indol-5-ylmethyl)amino]propanamide
(1-{7-methanesulfonyl-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-yl)methanol
1-{3,5-dimethyl-4-[3-(4-methylpyridin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrrol-2-yl}ethan-1-one
1-(pyrrolidine-1-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
methyl 2-[butyl(methyl)sulfamoyl]-6-[(3-chlorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(pyridin-4-ylmethyl)-4-[4-(2,2,2-trifluoroethyl)piperazine-1-carbonyl]pyrrolidin-2-one
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
2-[3-(dimethylamino)pyrrolidin-1-yl]-1-[3-(3-methoxyphenoxy)azetidin-1-yl]ethan-1-one
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-1-[(4-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-(3-cyclopentylpropanoyl)-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
methyl 4-(4-methyl-2-oxo-2H-chromen-7-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
1-cyclohexyl-4-(2-hydroxy-5-methoxyphenyl)-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1-phenylpyrrolidine-3-carboxamide
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(1-methylpiperidin-4-yl)piperidin-3-yl]propanoate
N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}-2-(naphthalen-1-yl)acetamide
2-({5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazol-3-yl}formamido)-N-cyclopropylacetamide
2-(4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
3-(furan-2-yl)-5-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}-1,2,4-oxadiazole
1-(2,3-dihydro-1H-inden-5-yl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
5-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
2-amino-6-(3,4-dichlorophenyl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
2-(3-methoxyphenyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
8-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
2-[2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethoxy]ethan-1-ol
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
1-{2-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-triene-5-carbonyl]phenyl}ethan-1-one
N-[(3S,4R)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-methyl-N-{1-[1-(4-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
3-(azepane-1-carbonyl)-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 1-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
(5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}furan-2-yl)methanol
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-2-(1H-indazol-1-yl)ethan-1-one
1-(2-ethyl-4-{[2-(oxolan-3-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)but-3-en-1-one
3-methyl-4-[3-phenyl-5-(1,2,3,6-tetrahydropyridin-4-ylmethyl)-1H-1,2,4-triazol-1-yl]pyridine
ethyl 1-[(4-methoxyphenyl)methyl]-5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-4-carboxamide
5-chloro-3-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-indole-2-carboxamide
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine