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(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanamine
3-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2,4-oxadiazole-5-carboxamide
2-{[5-(2,6-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methyl-1,3,4-oxadiazole
2-(1H-indol-3-yl)-N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
3-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
4-[(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-2-yl)methyl]morpholine
1-(2-{[(6-methoxypyridin-3-yl)methyl](methyl)amino}ethyl)piperidin-2-one
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[1-(methoxymethyl)cyclobutyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
2-(2-hydroxyethyl)-9-(4-methoxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(cyclopropylmethyl)-3-[(5-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
N,N-dimethyl-5-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-amine
methyl 2-(azepane-1-sulfonyl)-6-[(2-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-methyl-6-(propan-2-yl)pyrimidine
3-(1,3-benzothiazol-2-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}propanamide
2-[2-(1H-indol-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 2-[methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]acetate
5-methyl-4-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
4-[2-(dimethylamino)ethyl]-11-({[4-(trifluoromethoxy)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
ethyl 1-(1-benzylpyrrolidin-3-yl)-4-(cyclopropylmethyl)piperidine-4-carboxylate
3-benzyl-4-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}morpholine
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-ethanesulfonamido-N,1-dimethyl-2-phenyl-N-[1-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-{[7-(methylsulfanyl)-2-oxo-1,2-dihydroquinolin-3-yl]methyl}piperidine-3-carboxamide
N-(1-methyl-1H-pyrazol-3-yl)-2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]acetamide
1-{1-[1-(1-benzofuran-5-carbonyl)piperidin-4-yl]ethyl}-4-methylpiperazine
N-butyl-N,5-dimethyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-cycloheptanecarbonyl-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(1R,2R,6S,7S)-4-[3-(2-methoxyphenyl)benzoyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-methyl-3-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[3-(2-methylphenoxy)propyl]urea
2-methyl-4-({4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazin-1-yl}methyl)phenol
3-(2-ethylbutyl)-8-(2-hydroxypropanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(1S,5R)-6-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-(2-methyl-1H-indol-3-yl)ethan-1-one
3-[(2R,3R,6R)-5-[(4-ethoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[3-(3,4-diethoxyphenyl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-methyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
6-{3-[2-(dimethylcarbamoyl)ethyl]piperidin-1-yl}pyridine-3-carboxylic acid
2,6,8-trimethyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]quinoline-4-carboxamide
4-(4-methyl-1,3-thiazol-2-yl)-1-[(4-methylphenyl)methyl]piperazin-2-one
N,1-dimethyl-N-[2-(oxan-2-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[3-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrazine-2-carbonitrile
(5-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}furan-2-yl)methanol
[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
(2S,3S)-2-[(5-methoxy-4-oxo-1,4-dihydropyridin-2-yl)formamido]-3-methylpentanamide
1-[(3-methoxyphenyl)methyl]-4-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-one