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1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(2-fluorophenyl)ethan-1-one
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]pyrrolidin-3-yl}benzoic acid
5-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
6-(3,3-diphenylpiperidine-1-carbonyl)piperazin-2-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
(2S,4R)-4-amino-N,N-diethyl-1-(2-phenylpyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(1H-pyrazol-1-yl)butanamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-(3-hydroxy-2,2-dimethylpropyl)propanamide
N-methyl-6-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-[5-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)-1-methyl-1H-pyrrol-3-yl]ethan-1-one
N-methyl-N-(pyrimidin-4-ylmethyl)-5-(trifluoromethyl)pyridin-2-amine
2-{2-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}-N,N-dimethylethane-1-sulfonamide
4-({1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)piperazin-2-one
N-(diphenylmethyl)-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1,8-dibenzyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(1H-imidazol-1-yl)butan-2-yl]-6,8-dimethyl-3,4-dihydroquinazolin-4-one
2-methoxy-N-(3-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)acetamide
2,4-dimethyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,3-thiazole
1-(2,2-dimethylpropyl)-4-({thieno[2,3-d]pyrimidin-4-yl}amino)pyrrolidin-2-one
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-6-methyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
5-tert-butyl-4-{[4-methyl-2,5-dioxo-4-(piperidin-4-yl)imidazolidin-1-yl]methyl}furan-2-carboxamide
3-{1-[(2S)-1-acetylpyrrolidine-2-carbonyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
3-[(3R,4S)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-(5-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridin-4-yl}-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl)acetic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-ethyl-1,3-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
4-(4-methyl-1H-imidazole-2-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,N-dimethyl-2-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1R,5S)-N-[2-(4-methoxyphenyl)phenyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
6-(4-methanesulfonylphenyl)pyrazine-2-carboxylic acid
1-{6-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridin-3-yl}ethan-1-one
1-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-2-(pyridin-2-yl)-1H-1,3-benzodiazole
2-amino-6-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}pyrimidin-4-ol
6,8-dimethyl-3-{[(1R,5S)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1,2-dihydroquinolin-2-one
4-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N-methyl-4-oxobutanamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
4-(4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
8-[6-(methoxymethyl)pyridine-2-carbonyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
(2H-1,3-benzodioxol-5-ylmethyl)(methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
3-(1H-1,3-benzodiazol-2-yl)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
2-[2-(dimethylamino)-2-(3-methylphenyl)acetamido]-2-methylpropanoic acid
N-[1-(4-chlorophenyl)cyclobutyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
2-[(3R,4S)-3-{2-[carbamoyl(methyl)amino]acetamido}-4-(propan-2-yl)pyrrolidin-1-yl]acetic acid
1-(oxan-4-yl)-3-(4-phenylbenzoyl)piperidine
1-[3-(pyridin-4-yl)-5-[2-(pyrrolidin-1-yl)phenyl]-1H-1,2,4-triazol-1-yl]butan-2-ol