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2-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(benzenesulfonyl)-1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]propan-1-one
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidin-2-amine
1-(2-methyl-1,4-oxazepan-4-yl)-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
4-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-N-methyl-1,3-thiazol-2-amine
methyl 3-{1-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperidin-4-yl}propanoate
5-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]-1-ethyl-1H-1,2,4-triazole
N-ethyl-3-(2-hydroxyphenyl)-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
(2S)-2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-hydroxypropanamide
2-(2-{[methyl(thian-4-yl)amino]methyl}-4-(pyridin-2-yl)phenoxy)acetic acid
4-hydroxy-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-cyclohexanecarbonyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}pyrrolidine-2-carboxamide
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-4-(2-oxopyrrolidin-1-yl)benzamide
5-[4-(pyrimidin-5-yl)phenyl]-1,3,4-thiadiazol-2-amine
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[1-(4-fluorophenyl)ethyl]amine
3-({4-[(1S,2S)-2-hydroxycyclohexyl]piperazin-1-yl}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
N-ethyl-N-(oxolan-2-ylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
2-{6-hydroxy-4-[2-(methylamino)pyrimidine-5-carbonyl]-1,4-diazepan-1-yl}acetic acid
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-2-ethyl-4-methyl-1,3-oxazole
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
3-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
2-methoxy-1-{1'-[2-(propan-2-ylsulfanyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
N-benzyl-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
2-[2-(pyridin-2-yl)ethyl]-8-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(morpholin-4-yl)ethyl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-methyl-2-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
4-(2-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-2-oxoethyl)-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
4-(naphthalen-2-yloxy)-1-(5-propylpyrimidin-4-yl)piperidine-4-carboxylic acid
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
3-{[(cyclopropylmethyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
methyl 6-[(4-ethylphenyl)methyl]-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(4-cyano-2,5-difluorophenyl)-1,3-dimethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decane-8-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(3-methylphenyl)piperidin-1-yl]propan-1-one
3-chloro-5-[1-ethyl-3-(3-fluorophenoxymethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-4-{1H-pyrrolo[2,3-c]pyridin-5-ylmethyl}piperazine
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-ethyl-1-[(1-methyl-1H-indol-5-yl)methyl]pyrrolidine-3-carboxamide
2-(azepane-1-carbonyl)-4-methyl-N-(propan-2-yl)aniline
1-[(2-butoxy-3-methoxyphenyl)methyl]-2,4-dimethyl-1,4-diazepane
N-butyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
2-methyl-4-phenyl-1-(thiophen-2-ylmethyl)piperazine
methyl (2S)-1-{2-[4-(4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
3-[(cyclopentylamino)methyl]-N,N,7-trimethylquinolin-2-amine