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5-ethoxy-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)furan-2-carboxamide
N-[2-hydroxy-2-(3-phenoxyphenyl)ethyl]-1-methylpiperidine-4-carboxamide
1-{4-[(3S,4R)-3-cyclopropyl-4-[(pyrimidin-2-yl)amino]pyrrolidine-1-carbonyl]piperidin-1-yl}ethan-1-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-methyl-N-(oxolan-3-yl)piperidine-4-carboxamide
2-(4-hydroxypiperidin-1-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
N-phenyl-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}[1-(thiophen-2-yl)propan-2-yl]amine
4-{1-[1-(6-ethylpyrimidin-4-yl)piperidin-4-yl]ethyl}morpholine
N-[(1-cycloheptanecarbonylpiperidin-3-yl)methyl]naphthalene-1-carboxamide
methyl 5-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-5-oxopentanoate
4-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-chloro-4-fluoro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
(1S,5R)-3-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
1-[2-oxo-2-(piperidin-1-yl)ethyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1,3-dimethyl-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[2-({2-phenylimidazo[1,2-a]pyridin-6-yl}formamido)ethyl]acetamide
N,N-diethyl-1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidin-3-amine
methyl 1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazole-4-carboxylate
3-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]-1-(2-methyl-1H-imidazole-4-carbonyl)piperidine
2-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-4-(pyrimidin-5-yl)phenol
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
4-{[(2-methoxyethyl)(thiophen-2-ylmethyl)amino]methyl}benzoic acid
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-(4H-1,2,4-triazol-4-yl)pyridine
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(oxan-4-yl)acetamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
5-methyl-1'-(3-methyl-1-benzothiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 4-(cyclopropylmethyl)-1-[4-(piperidin-1-yl)benzoyl]piperidine-4-carboxylate
N-benzyl-5-cyclohexaneamido-N-(cyclopropylmethyl)-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
9-[(4-acetylphenyl)methyl]-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[1-(naphthalene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]pyrrolidin-3-amine
2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-6-methylpyrimidine-4-carboxamide
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
(3R)-1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
3-benzyl-1-methyl-3-{2-[4-(methylamino)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-indol-2-one
{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
(1-benzothiophen-2-ylmethyl)({4-[2-(4-{imidazo[1,2-a]pyridine-2-carbonyl}piperazin-1-yl)ethoxy]phenyl}methyl)methylamine
N-methyl-N-(1,3-thiazol-2-ylmethyl)-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
(1R,5R)-3-cyclobutanecarbonyl-6-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-(1H-1,2,3-benzotriazol-1-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
1-[(2-methoxy-3,5-dimethylphenyl)methyl]azetidine-2-carboxylic acid
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
N-(oxan-2-ylmethyl)-2-(pyridin-4-ylsulfanyl)acetamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
2-ethyl-N-[(8-methoxyquinolin-5-yl)methyl]-N,4-dimethyl-1,3-oxazole-5-carboxamide
1-{4-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]thiophen-2-yl}ethan-1-one
N-benzyl-N-methyl-3-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]benzamide