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3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
1-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carbonyl}piperidine-4-carbonitrile
2-hydroxy-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethan-1-one
methyl 4-[({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]benzoate
{5-fluoro-2-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}methanamine
N-{[4-(cyclooctyloxy)phenyl]methyl}-4-acetamido-N-(pyridin-3-ylmethyl)benzamide
N-benzyl-2-[4-(4-{[1-(thiophen-2-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide
2-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
N-[(4-chlorophenyl)(phenyl)methyl]-1-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carboxamide
7-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(3R,4S)-4-cyclopropyl-1-[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)benzenesulfonyl]pyrrolidin-3-amine
5-cyclopropanecarbonyl-1'-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-methyl-3-[4-(2-oxopyrrolidin-1-yl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-(propan-2-yloxy)propan-1-one
3-({1-[3-(4H-1,2,4-triazol-4-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(2-fluorophenyl)-3-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
1-(2-methylpropyl)-5-(morpholin-4-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
3-[4-(2-fluorophenyl)-1H-pyrazol-5-yl]-1-(2-phenylpropyl)piperidine
2,6-dimethyl-3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]quinoline
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
N-[2-(4-fluorophenyl)-1-(1-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}piperidin-4-yl)ethyl]-2-methoxy-N-methylacetamide
2,6-diamino-4-cyclopropyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
4-methyl-9-(1-phenyl-1H-pyrazol-5-yl)-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
2-(3-{3-[5-(trifluoromethyl)pyridin-2-yl]phenyl}-1H-pyrazol-1-yl)acetamide
4-(1H-pyrazol-3-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide
4-(1-ethyl-1H-imidazol-2-yl)-1-[(4-methanesulfonylphenyl)methyl]piperidine
N-methyl-2-(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-(1H-1,3-benzodiazol-2-ylmethyl)-N-cyclopentyl-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{1-[1-(furan-3-ylmethyl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-3-ylmethyl)amine
2-methyl-3-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1H-indol-4-one
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(2-{methyl[(4-methylphenyl)methyl]amino}acetamido)acetic acid
N,N-diethyl-1-[1-(2-methyl-2-phenylpropanoyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
(3S,5R)-N5-(2,3-dihydro-1H-inden-5-yl)-N3,N3-dimethyl-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
2-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-6-methyl-1H-1,3-benzodiazole
N-[(6-chloro-2H-chromen-3-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
(2R,6R)-4-cyclobutanecarbonyl-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
8-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-methyl-5-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrole-3-carbonitrile
5-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenoxy}-1-azabicyclo[3.2.1]octane
ethyl 1-(2-methylpropyl)-5-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(2-tert-butylpyrimidin-5-yl)-N,8-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
N-(3-carbamoylphenyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
N-cyclopropyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
2-chloro-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
(1S,5R)-6-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(3-methylpyridin-2-yl)methyl]-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one