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9-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(oxane-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]-N-(dimethyl-1,2-oxazol-4-yl)piperidine-1-carboxamide
[(3R,4R)-1-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
6-[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-2-carbonitrile
N-(2,2-dimethyloxan-4-yl)-5-methanesulfonamido-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
2-[3-(5-chloro-2-ethoxyphenyl)phenoxy]acetamide
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(2-methoxyphenyl)methyl]piperidin-4-ol
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-(1H-pyrazol-4-yl)propan-1-one
1-[1-(pyridazine-3-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
3-(2-{1',5',6',7'-tetrahydrospiro[cyclohexane-1,4'-imidazo[4,5-c]pyridine]-5'-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
5-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
N,4-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-6H,7H,8H-cyclopenta[g]quinazolin-2-amine
(1R,5R)-6-(2,5-dimethylfuran-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
1-ethyl-5-{1-[2-(2-methoxyphenyl)ethyl]-4-phenyl-1H-imidazol-5-yl}-1H-1,2,4-triazole
4-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-5-propylpyrimidine
1-({5-[(3-ethenylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-cyclopropyl-8-[4-(ethylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
5-(1H-imidazol-2-yl)-2-(naphthalen-1-yl)pyrimidine
7-(5-acetylthiophene-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[2-(pyridin-3-yloxy)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[2-(prop-2-en-1-yloxy)phenyl]methyl})(pyridin-4-ylmethyl)amine
5-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-(2-methoxyethyl)-N-(naphthalen-1-ylmethyl)acetamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-3-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}piperidine
1-benzyl-N-{7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidin-3-amine
1-[4-({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)-1,4-diazepan-1-yl]ethan-1-one
4-[4-(4-methylphenoxy)piperidine-1-carbonyl]pyridin-2-amine
1-[(3R,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]naphthalen-2-ol
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5,8-dimethoxy-4-methylquinoline
8-[(4-chlorophenyl)methyl]-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
2-[5-(2,3-difluoro-6-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]-2-ethylpropane-1,3-diol
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]acetamide
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-5-methoxy-3-methyl-1H-indole
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
1-[(3,4-dimethylphenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-2-one
2-(4-fluorophenyl)-N-[2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)ethyl]acetamide
2-[2-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-{phenyl[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
methyl 1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]cyclopropane-1-carboxylate
N-(cyclohex-1-en-1-ylmethyl)-2-(4-{2-[4-(dimethylamino)phenyl]acetyl}morpholin-3-yl)acetamide
(3S,9aR)-8-(3-chlorobenzoyl)-3-(cyclohexylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{imidazo[1,2-a]pyridin-2-yl}-5-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1,2,4-oxadiazole
2-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-5-ol
5-methyl-3-{3-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1,3-benzoxazol-2-one
N,2,5-trimethyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine