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1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(morpholin-4-yl)ethan-1-one
8-(isoquinolin-1-yloxy)-5-(morpholin-4-ylmethyl)quinoline
2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]pyridine-4-carboxylic acid
4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
2-(2-{methyl[2-(morpholin-4-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[4-methyl-2-(2-{[methyl(propan-2-yl)amino]methyl}propanamido)phenyl]pentanamide
dimethyl(3-{2-[1-(5,6,7,8-tetrahydroquinolin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
2-(2-ethyl-1H-imidazol-1-yl)-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
(2S,3R)-2-amino-3-hydroxy-1-[4-(2-methylphenoxy)piperidin-1-yl]butan-1-one
1-({5-[1-(2-hydroxyethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-2-(propan-2-yl)pyrimidine
2-(3,4-dimethoxyphenyl)-4-[3-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
methyl (2S,4R)-4-[3-(4-methylphenyl)propanamido]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-5-(methoxymethyl)thiophene-2-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(1R,5R)-6-{[3-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-(2-acetamidoethyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-[(2-fluorophenyl)methyl]-N-[(6-methylpyridin-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-methylacetamide
5-[(dimethylsulfamoyl)amino]-1-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(2-butyl-1H-imidazol-4-yl)methyl](ethyl)({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amine
3-(2-amino-1,3-thiazol-4-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N-{4-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl}methanesulfonamide
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(2-ethoxyethyl)-1,4-diazepan-6-ol
methyl 1-(2-methoxyethoxy)-2-oxo-8-(4-phenylbenzoyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(3-chlorophenyl)-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}propanoic acid
3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-2,8-diazaspiro[4.5]decane
4-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]benzoic acid
N-(2,3-difluorophenyl)-2-(2-methoxyethyl)morpholine-4-carboxamide
[(3R,4R)-1-(5-chloro-2-methylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
6-[3-(2-methoxyphenyl)propanoyl]-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-fluorophenyl)ethyl]acetamide
(3S,4S)-4-(dimethylamino)-1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-ol
2-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}pyrazine
1-[4-(3-{[(quinolin-2-yl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-(1-methoxypropan-2-yl)piperidine-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
3-(1,3-dimethyl-1H-pyrazol-5-yl)-1-{[1-(3-fluorophenyl)cyclopentyl]methyl}urea
2-[(3,4-difluorophenyl)methyl]-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
(2S,3R)-2-amino-1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-hydroxybutan-1-one
methyl 4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carboxylate
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-phenylacetamide
2-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
5-[1-(5-methyl-2-phenylfuran-3-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
(1S,5R)-3-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-({[4-methyl-3-(2-oxoimidazolidin-1-yl)phenyl]formamido}methyl)-1,2,4-oxadiazole-5-carboxamide
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-1-methylurea