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1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(1-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyrazine
4-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-1,4-diazepane-1-carbaldehyde
N3-ethyl-N5-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(2S)-2-{[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido}-3-(pyridin-4-yl)propanoic acid
ethyl 4-[(2-chlorophenyl)methyl]-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidine-4-carboxylate
2-{[1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}benzamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methylpiperidine-4-carbonyl)piperidine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-(furan-3-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-ethyl-5-({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-butyl-N-cycloheptyl-2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]acetamide
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(2-phenoxyethyl)acetamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-5-(1H-imidazol-1-ylmethyl)furan-2-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)benzamide
1-[2-({[4-(ethylcarbamoyl)-2-methylphenyl]carbamoyl}amino)ethyl]piperidine-3-carboxamide
4-(cyclopropylmethyl)-N-[4-(ethylsulfanyl)phenyl]-3-(2-hydroxyethyl)piperazine-1-carboxamide
1-(3-methoxyphenyl)-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-2-one
(benzylsulfamoyl)(ethyl)[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amine
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-(4-methoxyphenyl)piperazin-2-one
2-({[3-(dimethylamino)phenyl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-(1,4-oxazepan-6-ylmethyl)-3-[4-(propan-2-yl)phenyl]urea
4-{5-[3-(2-methylpropyl)-1,2-oxazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridine
N-(3-methoxypropyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-(2,3-difluorophenyl)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}ethan-1-one
N-cyclohexyl-N-methyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
1-cyclobutanecarbonyl-N-(4-fluorophenyl)piperidin-3-amine
2-(4-methoxyphenoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
1-cyclohexyl-3-methyl-5-(1-methyl-1H-pyrrol-2-yl)-1H-1,2,4-triazole
N-cyclohexyl-2-[(3R,4S)-3-acetamido-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]acetamide
4-(2-methoxyphenyl)-3-(2-phenylethyl)-4H-1,2,4-triazole
6-ethyl-2-methyl-N-[3-(methylsulfanyl)propyl]quinoline-4-carboxamide
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-4-hydroxy-1-methylpiperidine-4-carboxamide
N-(1H-1,3-benzodiazol-2-yl)-2-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]amino}acetamide
2-methyl-5-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)-1,4-dihydropyridin-4-one
N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
(4aS,8aR)-1-[(5-methylfuran-2-yl)methyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(3,5-dimethylphenyl)propan-1-one
2-{[(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)oxy]methyl}pyridine
[(3aS,6aS)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-3-(pyridin-3-yl)propan-1-one
N-ethyl-4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-amido]piperidine-1-carboxamide
(3aS,6aS)-2-methyl-5-[2-methyl-5-(1H-pyrazol-1-yl)benzenesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
6-[2-(benzyloxy)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile