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2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
methyl 3-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
3-cyclopropyl-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
2-methyl-4-[1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-3-yl]-6-(pyrrolidin-1-yl)pyrimidine
(2S)-N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methylpyrrolidine-2-carboxamide
{2-[5-chloro-2-(propan-2-yloxy)phenyl]pyridin-4-yl}methanol
2-(6-methoxynaphthalen-2-yl)-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
N-methyl-N-[2-(phenylsulfanyl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-4,6-dioxo-3-[2-(1H-pyrazol-1-ylmethyl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(1-methylcyclopropanecarbonyl)-3-[2-(2-methylphenyl)ethyl]piperidine
4-[(dipropylamino)methyl]-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-[(3-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-oxazol-5-yl)methyl]piperidin-4-ol
N-[2-(diethylamino)ethyl]-N-methyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-(1H-imidazol-1-yl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
2-cyclohexyl-6-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1,3-benzoxazole
N-(9H-fluoren-9-yl)-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(2-methoxyphenyl)-1H-indazol-1-yl]acetamide
2-amino-6-{4-[(dimethylamino)methyl]thiophen-2-yl}-4-(1-ethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-ethyl-6-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
3-{[1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperidin-4-yl]methyl}benzoic acid
3-(3-methoxypropyl)-N-(4-phenoxyphenyl)piperidine-1-carboxamide
4-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-6-methylpyrimidin-2-amine
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}butan-1-one
2-{4-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}-N-(1-ethyl-1H-pyrazol-5-yl)acetamide
N,2-dimethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(5-methoxypyridin-3-yl)-N,N-dimethylthiophene-2-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-methyl-1-(2-phenylethyl)-N-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-amine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-2-fluoro-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-2-ylmethyl)pyridin-2-amine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[3-(1H-indazol-1-yl)propyl]acetamide
2-{4-[(6-hydroxy-1,4-oxazepan-4-yl)methyl]phenyl}acetic acid
5-methyl-5-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
2-hydroxy-4-methyl-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pentan-1-one
1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)piperidine-2-carboxamide
7-[3-(5-methylfuran-2-yl)butyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-butyl-5-phenyl-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-ethyl-3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-pyrazole
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
4-benzyl-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-3-ethyl-1,4-diazepan-5-one
1-methyl-N-(2-phenoxyethyl)-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(2S,4S)-4-amino-N-ethyl-1-(4-hydroxy-6-oxo-1-phenyl-1,6-dihydropyridazine-3-carbonyl)pyrrolidine-2-carboxamide
2-(3-methylphenyl)-5-{1-[2-(piperidin-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
N-[(3-chlorophenyl)methyl]-3-[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]propanamide