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1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N5-cyclopentyl-N6-(2,2-dimethyloxan-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(3-methyl-1,2-oxazol-5-yl)-N-propyl-N-(pyridin-3-ylmethyl)acetamide
1-[2-(3,4-difluorophenyl)acetyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-[2-(2-fluorophenyl)ethyl]-5-{1-[(4-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-1-benzofuran-2-carboxamide
(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-amine
(2S,4S)-4-amino-N-methyl-1-(1-propyl-1H-pyrazole-5-carbonyl)pyrrolidine-2-carboxamide
5-{2H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]benzamide
6-(2-hydroxyethyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(propan-2-yl)-1-(2-{4-[2-(trifluoromethyl)benzenesulfonyl]piperazin-1-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N1,N1-dimethyl-N4-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1,4-dicarboxamide
N-(3,4-dimethylphenyl)-1-(1-methyl-1H-indole-3-carbonyl)piperidin-3-amine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-methyl-5-phenyl-1H-pyrrole-2-carboxamide
3-({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)sulfamoyl)-N,N-dimethylbenzamide
3-(4-hydroxyphenyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
N-[3-(1H-indol-1-yl)propyl]-2-(pyrrolidin-3-yl)acetamide
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-5-phenyl-1,2-oxazole-3-carboxamide
2-(4-fluorophenoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
4-(3-acetylbenzoyl)-1-(3-chlorophenyl)-5-methylpiperazin-2-one
(3R,9aR)-8-(4-chlorobenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2,6-dimethyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}pyrimidine-4-carboxamide
(1R,2R,4R)-N-[2-(1H-indol-1-yl)ethyl]-N-methylbicyclo[2.2.1]hept-5-ene-2-carboxamide
(1R,3S)-3-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}cyclopentan-1-amine
9-(2-phenylethyl)-3-oxa-9-azaspiro[5.5]undecane
2-methyl-8-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-2,8-diazaspiro[4.5]decane
(3R,5S)-N-[3-(dimethylamino)propyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl](oxolan-2-ylmethyl)amine
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
(2S,4S)-4-amino-1-(3-cyanobenzenesulfonyl)-N,N-diethylpyrrolidine-2-carboxamide
3-ethyl-1-[4-(2-hydroxyphenyl)phenyl]urea
2-ethoxy-5-{2-[3-(hydroxymethyl)piperidin-1-yl]pyrimidin-4-yl}benzoic acid
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(2-methoxyacetamido)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 5-(cyclobutylamino)-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[(5-chlorofuran-2-yl)methyl]-1-phenylpiperazin-2-one
N-{3-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-oxopropyl}-4-fluorobenzamide
5-hydroxy-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}pyrazine-2-carboxamide
3-{[4-methyl-6-(3-phenylpiperazin-1-yl)pyrimidin-2-yl]amino}phenol
1-ethyl-4-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
(3R,4S)-1-(3-chloro-4-fluorobenzoyl)-3,4-dimethylpiperidin-4-ol
ethyl 2-[1-(2-butyl-1,3-benzoxazole-5-carbonyl)piperidin-2-yl]acetate
2-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-1H-1,3-benzodiazole-5-carbonitrile
N-(3-carbamoylphenyl)-3-{[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]methyl}benzamide
N-[(1R,2S)-2-phenylcyclohexyl]-2-(piperidin-4-yl)acetamide
dimethyl({5-[(2-phenylazetidin-1-yl)methyl]thiophen-3-yl}methyl)amine
methyl(2-phenylethyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N-ethyl-N-methyl-3-{methyl[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]sulfamoyl}benzamide
methyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
1'-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]