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1-(4-methoxyphenyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]cyclopropane-1-carboxamide
3,5-dimethyl-1-[1-(1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]-1H-pyrazole
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
5-[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
(2R,6R)-4-cyclopropanecarbonyl-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[4-(2-fluoro-5-methylphenyl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-N-methylacetamide
4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)piperidine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(1,3-oxazol-5-yl)phenyl]pyrrolidine-1-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-(piperidin-1-yl)-1-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
N-(2,2-difluoroethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-{2-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]pyridin-3-yl}-2-methylpropanamide
1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
N-ethyl-N-[(5-methylfuran-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1'-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-(2-fluorophenoxymethyl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-ethylpyridine-4-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(2-methoxypyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{2,3-dimethyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
N-(propan-2-yl)-2-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-amine
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-[(3-methylphenyl)methyl]piperazine
2-(2-chloropyridine-4-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-{[6-(8-methoxy-2-methylquinolin-5-yl)pyridazin-3-yl]amino}ethan-1-ol
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-2-one
8-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-(4-acetyl-1,4-diazepan-1-yl)-3-(4-methoxyphenyl)-3-phenylpropan-1-one
4-(6-{octahydropyrrolo[1,2-a]piperazin-2-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl)morpholine
2-[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
7-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-1H-indole
2-{2-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
6-methoxy-2-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
2-[3-(4-fluorophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-[(2-fluorophenyl)methyl]-5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(1S,5R)-3-[(2-methoxynaphthalen-1-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxyethyl)-2-methyl-N-(thiophen-2-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(1S,3R)-3-[1-ethyl-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]-N,2,2,3-tetramethylcyclopentane-1-carboxamide
N,N-dimethyl-4-[3-(thiomorpholine-4-carbonyl)phenoxy]piperidine-1-sulfonamide
4-[2-(2-chloro-6-fluorophenyl)acetyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
{3-[(3-chlorophenyl)methyl]-1-(1,4-dithiepan-6-yl)piperidin-3-yl}methanol
3-benzyl-1-methyl-8-{[4-(methylsulfanyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(cyclopropylmethyl)-4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(propan-2-yl)-1,4-diazepane
N-(furan-2-ylmethyl)-3,5-dimethoxy-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
(3R,4S)-4-cyclopropyl-1-[3-(trifluoromethyl)benzenesulfonyl]pyrrolidin-3-amine
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(6-methoxyquinolin-8-yl)-3-methylurea
(2R,3R,6R)-3-(4-methylphenyl)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl (2R,4S)-4-hydroxy-1-[(4-methyl-3,4-dihydro-2H-1,4-benzoxazin-7-yl)sulfonyl]piperidine-2-carboxylate
1-[4-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one