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1-[5-(methoxymethyl)furan-2-carbonyl]-3-(3-methylphenoxymethyl)piperidine
methyl 2-(1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}-N-methylformamido)acetate
N-cyclopropyl-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-3-methylthiophene-2-carboxamide
1-({3-[(2S,5R)-2,5-dimethylpiperazine-1-carbonyl]-1,2-oxazol-5-yl}methyl)-2-methyl-1H-1,3-benzodiazole
ethyl 4-{1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carbonyl}piperazine-1-carboxylate
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-methyloxolane-2-carboxamide
3,3-dimethyl-1-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}urea
N,N-dimethyl-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}aniline
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidin-3-yl]methanol
methyl 3-cyclohexyl-1-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
{1-[(4,5-dimethylfuran-2-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
(5-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}-2-(propan-2-yloxy)phenyl)methanol
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(1H-imidazol-1-yl)propan-1-one
3-(1-propyl-1H-pyrazol-5-yl)-1-[1-(thiophen-3-yl)propan-2-yl]urea
2-cyclopropyl-4-phenyl-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane
N-butyl-5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
5-{[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
11-(benzylamino)-4-(3-methoxypropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
6-(methoxymethyl)-N-{2-[2-(propan-2-yloxy)phenyl]ethyl}pyrimidin-4-amine
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(3-methoxypropyl)acetamide
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-methyl-1,3-oxazole-4-carboxamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-(5,6-dimethylpyrimidin-4-yl)-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
2-{[4-(1-phenylethyl)-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(2-methoxyphenyl)-3-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}urea
N,2-dimethyl-N-(1,2-oxazol-3-ylmethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
methyl 2-[3-(2-methyl-1H-indol-1-yl)propanamido]-4-(methylsulfanyl)butanoate
1-(3-methoxypiperidin-1-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
2-(methylsulfanyl)-4-{4-[4-(oxolan-2-ylmethyl)piperazin-1-yl]piperidin-1-yl}pyrimidine
3-[(dimethylamino)methyl]-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-{[4-(hydroxymethyl)phenyl]methyl}acetamide
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
(3-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-6-methoxyphenol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-ethoxy-N-(oxolan-2-ylmethyl)acetamide
5-chloro-2-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
1-{2-[3-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}piperidine-2,6-dione
1-(2,3-dihydro-1H-inden-2-yl)-5-(2-methyl-1H-pyrrol-3-yl)-1H-1,2,4-triazole
3,6,7-trimethyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-benzofuran-2-carboxamide
(4aR,7aS)-1-{2-[butyl(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[3-methyl-7-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-8-fluoro-N-methylquinoline-2-carboxamide
2-{[4-(3-fluorophenoxy)piperidin-1-yl]methyl}-6-methylpyridine
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
(4S)-4-acetamido-4-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]butanamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[(2,4,6-trimethylphenyl)methyl]urea
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine