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3-(2-methoxyethyl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine-3-carboxylic acid
1-{4-[({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]piperidin-1-yl}-2-methylpropan-1-one
2-[4-(3-cyanophenyl)phenyl]-N,N-dimethylacetamide
2-{5-[1-(3,4-difluorobenzoyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
6-cyclopentyl-N,1-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[(3-methyl-1H-pyrazol-4-yl)methyl]amine
5-acetyl-2,4-dimethyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-pyrrole-3-carboxamide
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-methyl-9-(1H-pyrazole-4-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
{2,4,6-trimethyl-3-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]phenyl}methyl acetate
6-[4-(7-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
1-cyclopentyl-4-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine
1-cyclobutanecarbonyl-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
6-(4-{[4-hydroxy-3-(prop-2-en-1-yl)phenyl]methyl}piperazin-1-yl)pyridine-3-carboxamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
2-ethoxy-4-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}phenol
2-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
(2S,4R)-4-[(adamantan-2-yl)amino]-1-[(2-chlorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(oxolane-2-carbonyl)piperidine
1-[(2-chlorophenyl)methyl]-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]-1,4-diazepan-5-one
6-(2-methanesulfonylphenyl)quinazolin-4-amine
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
2-[(3Z)-hex-3-en-1-yl]-1H-1,3-benzodiazole
2-hydroxy-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
4'-[(4,6-dimethylpyrimidin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-cyclopentylpiperidin-2-one
N-[2-(benzylsulfanyl)ethyl]-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
1-[3-(3-ethylphenoxy)azetidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-cyclobutaneamido-N-[(3-methyl-1H-pyrazol-5-yl)methyl]benzamide
3-{1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}piperidine
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-benzyl-3-cyclopropyl-5-[(4-methanesulfonylphenyl)methyl]-1H-1,2,4-triazole
({4-cyclopropyl-5-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-(2-methyl-1H-imidazol-1-yl)-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]propan-1-one
5-(4-methoxy-2,3-dimethylphenyl)-1-(oxan-4-yl)-4-phenyl-1H-imidazole
2-cyclopropanecarbonyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-{4-[1-(dimethylamino)ethyl]phenyl}-N,N-dimethylbenzamide
1-(2-chlorophenyl)-3-{1-[1-(pent-4-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
(2S,4R)-N-cyclopropyl-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
(1S,5R)-6-{[4-(methylsulfanyl)phenyl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperidin-4-yl]pyridine
3-({[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-N-(pyridin-4-yl)benzamide
1-cyclopentyl-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
8-[(6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
1-(diethylamino)-3-[4-({[(2,6-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol